SCHEMBL4553447

SCHEMBL4553447

CC(C)(C)OC(=O)Cn1cc(-c2ccc(Br)cc2)nn1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SRC P12931 5/20 0.49
NR1H4 Q96RI1 1/20 0.46
BCL2L11 O43521 1/20 0.45
BCL2L1 Q07817 1/20 0.45
MCL1 Q07820 1/20 0.45
HSP90AA1 P07900 2/20 0.41
HSP90AB1 P08238 2/20 0.41
HDAC3 O15379 3/20 0.41
HDAC4 P56524 3/20 0.41
HDAC1 Q13547 3/20 0.41
HDAC7 Q8WUI4 3/20 0.41
HDAC2 Q92769 3/20 0.41
HDAC10 Q969S8 3/20 0.41
HDAC11 Q96DB2 3/20 0.41
HDAC8 Q9BY41 3/20 0.41
HDAC6 Q9UBN7 3/20 0.41
HDAC9 Q9UKV0 3/20 0.41
HDAC5 Q9UQL6 3/20 0.41
DRD2 P14416 1/20 0.41
DRD4 P21917 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14140577 0.80 NPC1 (0.56) MEN1NPC1RAB9AKMT2A
SCHEMBL4552469 0.80 NPC1 (0.56) MEN1NPC1RAB9AKMT2A
SCHEMBL25170515 0.78 KCNH2 (0.45) HDAC3HDAC8
SCHEMBL4553061 0.76 FFAR1 (0.41) SRCNR1H4BCL2L11BCL2L1MCL1
SCHEMBL26454236 0.76 CCNC (0.41) HDAC6NPC1RAB9A
SCHEMBL22576897 0.75 ALDH1A1 (0.38) SRCNR1H4BCL2L11BCL2L1MCL1
SCHEMBL5053636 0.73 CYP19A1 (0.45) SRCNR1H4HSP90AA1HSP90AB1HDAC3
SCHEMBL28497312 0.72 MITF (0.39) SRCBCL2L11BCL2L1MCL1HDAC6
SCHEMBL22958957 0.72 SRC (0.52) SRCHDAC3HDAC4HDAC1HDAC7
SCHEMBL22959003 0.71 SRC (0.58) SRCHDAC3HDAC4HDAC1HDAC7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101610674-A Sphingosine-1-phosphate ester receptor stimulating agent and agonist compounds ABBOTT LAB (US) 2009-12-23 CN disclosed
EP-2120575-A1 SPHINGOSINE-1 -PHOSPHATE RECEPTOR AGONIST AND ANTAGONIST COMPOUNDS Abbott Laboratories (US) 2009-11-25 EP disclosed
WO-2008079382-A1 SPHINGOSINE-1 -PHOSPHATE RECEPTOR AGONIST AND ANTAGONIST COMPOUNDS ABBOTT LABORATORIES (US) 2008-07-03 WO disclosed
WO-2008079382-A1 SPHINGOSINE-1 -PHOSPHATE RECEPTOR AGONIST AND ANTAGONIST COMPOUNDS ABBOTT LABORATORIES (US) 2008-07-03 WO disclosed