SCHEMBL4554664

SCHEMBL4554664

O=C(O)NC[C@@H]1OC(=O)N2c3ccc(C4=CC[S+]([O-])CC4)cc3C[C@@H]12

nearest known ligand 0.35

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 0.35
F10 P00742 18/20 0.34
MAOA P21397 1/20 0.32
MAOB P27338 1/20 0.32
CYP2C19 P33261 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9930084 0.92 KCNH2 (0.43) KCNH2F10MAOAMAOBCYP2C19
SCHEMBL9930468 0.84
SCHEMBL4555333 0.82 MAOA (0.38) KCNH2F10MAOAMAOBCYP2C19
SCHEMBL9930612 0.81 MAOA (0.34) KCNH2MAOAMAOB
SCHEMBL9964815 0.76 KCNH2 (0.46) KCNH2F10MAOAMAOBCYP2C19
SCHEMBL4555076 0.74 MAOA (0.47) KCNH2F10MAOAMAOBCYP2C19
SCHEMBL9929840 0.74 MAOA (0.46) KCNH2F10MAOAMAOBCYP2C19
SCHEMBL9930383 0.72 KCNH2 (0.42) KCNH2F10MAOAMAOBCYP2C19
SCHEMBL9930417 0.70 MAOA (0.42) KCNH2F10MAOAMAOBCYP2C19
SCHEMBL9930581 0.70 NAMPT (0.44) KCNH2F10MAOAMAOBCYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2134721-A1 ANTIMICROBIAL HETEROCYCLIC COMPOUNDS FOR TREATMENT OF BACTERIAL INFECTIONS Micurx Pharmaceuticals, Inc. (US) 2009-12-23 EP disclosed
WO-2008108988-A1 ANTIMICROBIAL HETEROCYCLIC COMPOUNDS FOR TREATMENT OF BACTERIAL INFECTIONS MICURX PHARMACEUTICALS, INC. (US) 2008-09-12 WO disclosed