SCHEMBL4554834

SCHEMBL4554834

COC(=O)C(Cc1ccc(C(=O)O)cc1)n1cc(CNc2ccc(S(N)(=O)=O)cc2)nn1

nearest known ligand 0.46

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CA2 P00918 13/20 0.46
CA1 P00915 12/20 0.46
CA12 O43570 10/20 0.46
CA9 Q16790 8/20 0.46
PTGS2 P35354 3/20 0.43
CA7 P43166 3/20 0.42
IL1RN P18510 1/20 0.41
ERAP2 Q6P179 1/20 0.41
PTPN2 P17706 1/20 0.41
PTPN1 P18031 1/20 0.41
CA14 Q9ULX7 1/20 0.40
ALDH1A1 P00352 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3743022 0.89 CA2 (0.49) CA2CA1CA12CA9CA14
SCHEMBL3729753 0.83 CA2 (0.56) CA2CA1CA12CA9PTGS2
SCHEMBL4555164 0.75 CA2 (0.54) CA2CA1CA12CA9CA7
SCHEMBL4553904 0.74 CA2 (0.48) CA2CA1CA12CA9CA7
SCHEMBL31675059 0.72 IL1RN (0.53) PTGS2IL1RNERAP2PTPN2PTPN1
SCHEMBL3743147 0.72 CA2 (0.49) CA2CA1CA12CA9PTGS2
SCHEMBL31675092 0.68 PTGS2 (0.49) CA2CA1CA12CA9PTGS2
SCHEMBL31675086 0.67 IL1RN (0.47) PTGS2IL1RNERAP2PTPN2PTPN1
SCHEMBL13012614 0.67 CA2 (0.62) CA2CA1CA12CA9PTGS2
SCHEMBL3736212 0.66 CA2 (0.48) CA2CA1CA12CA9CA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2129666-A2 DEVELOPMENT OF MOLECULAR IMAGING PROBES FOR CARBONIC ANHYDRASE-IX USING CLICK CHEMISTRY Siemens Medical Solutions USA, Inc. (US) 2009-12-09 EP claimed
WO-2008124703-A2 DEVELOPMENT OF MOLECULAR IMAGING PROBES FOR CARBONIC ANHYDRASE-IX USING CLICK CHEMISTRY SIEMENS MEDICAL SOLUTIONS USA, INC. (US) 2008-10-16 WO claimed
EP-2129666-A2 DEVELOPMENT OF MOLECULAR IMAGING PROBES FOR CARBONIC ANHYDRASE-IX USING CLICK CHEMISTRY Siemens Medical Solutions USA, Inc. (US) 2009-12-09 EP disclosed
WO-2008124703-A2 DEVELOPMENT OF MOLECULAR IMAGING PROBES FOR CARBONIC ANHYDRASE-IX USING CLICK CHEMISTRY SIEMENS MEDICAL SOLUTIONS USA, INC. (US) 2008-10-16 WO disclosed