SCHEMBL4555245

SCHEMBL4555245

O=S(=O)(c1ccccc1)n1cc(I)cc1C1CCCCC1

nearest known ligand 0.44

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 8/20 0.44
ALDH1A1 P00352 3/20 0.43
ACHE P22303 1/20 0.40
KDM4E B2RXH2 1/20 0.40
GAA P10253 1/20 0.40
LMNA P02545 2/20 0.38
HTT P42858 1/20 0.38
TSHR P16473 1/20 0.37
PARL Q9H300 1/20 0.37
EPHX2 P34913 1/20 0.37
NPC1 O15118 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1156431 0.81 HTR6 (0.43) HTR6ALDH1A1ACHEKDM4EGAA
SCHEMBL1580856 0.77 HTR6 (0.40) HTR6ALDH1A1ACHEEPHX2
Hydrochloric Acid SCHEMBL1156400 0.76 HTR6 (0.39) HTR6ALDH1A1ACHEKDM4EEPHX2
SCHEMBL1156305 0.74 MAPK1 (0.47) ALDH1A1HTTNPC1
SCHEMBL1156715 0.73 ACHE (0.41) HTR6ALDH1A1ACHEKDM4ELMNA
SCHEMBL1799962 0.70 BRD4 (0.54) HTR6ALDH1A1KDM4ELMNAHTT
SCHEMBL1580453 0.69 HTR6 (0.41) HTR6ALDH1A1ACHEKDM4E
Hydrochloric Acid SCHEMBL1156630 0.69 HTR6 (0.41) HTR6ALDH1A1ACHEKDM4E
SCHEMBL1156354 0.69 KMT2A (0.49) ALDH1A1KDM4EGAALMNATSHR
SCHEMBL29065523 0.67 HTR6 (0.38) HTR6ALDH1A1KDM4EPARL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2125801-A1 THE USE OF 7-AZAINDOLES IN THE INHIBITION OF C-JUN N-TERMINAL KINASE Eisai R&D Management Co., Ltd. (JP) 2009-12-02 EP disclosed
WO-2008095943-A1 THE USE OF 7-AZAINDOLES IN THE INHIBITION OF C-JUN N-TERMINAL KINASE EISAI R&D MANAGEMENT CO. LTD. (JP) 2008-08-14 WO disclosed