SCHEMBL4556057

SCHEMBL4556057

O=C(O)N1CCC(Oc2cccc3ccc(Cl)nc23)C(F)C1

nearest known ligand 0.40

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
PIM1 P11309 13/20 0.40
PIM2 Q9P1W9 13/20 0.40
MCHR1 Q99705 7/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL731935 0.86 SMN1; SMN2 (0.43) MCHR1
SCHEMBL731934 0.86 SMN1; SMN2 (0.43) MCHR1
SCHEMBL4446931 0.85 KDM4E (0.48)
SCHEMBL17443063 0.75 KCNH2 (0.39)
SCHEMBL8515681 0.74 LPL (0.44)
SCHEMBL5884467 0.73 MCHR1 (0.65) MCHR1
SCHEMBL731475 0.72 KDR (0.49) PIM1PIM2
SCHEMBL729951 0.71 GPR119 (0.44)
SCHEMBL729950 0.71 GPR119 (0.44)
SCHEMBL731052 0.71 GRIN2B (0.47)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2137184-A1 IMIDAZO[1,2-A]PYRIDINE COMPOUNDS AS RECEPTOR TYROSINE KINASE INHIBITORS Array Biopharma, Inc. (US) 2009-12-30 EP disclosed
WO-2008124323-A1 IMIDAZO[1,2-A]PYRIDINE COMPOUNDS AS RECEPTOR TYROSINE KINASE INHIBITORS ARRAY BIOPHARMA INC. (US) 2008-10-16 WO disclosed