SCHEMBL4556732

SCHEMBL4556732

CC(C)(C)OC(=O)N1CCCc2c(O)cccc21.CC(C)(C)OC(=O)N1CCCc2c1ccc(Cl)c2O

nearest known ligand 0.41

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
UCHL1 P09936 3/20 0.41
HDAC1 Q13547 1/20 0.40
HDAC6 Q9UBN7 1/20 0.40
NOTUM Q6P988 4/20 0.38
KDM1A O60341 1/20 0.38
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
GPR119 Q8TDV5 1/20 0.36
BRD4 O60885 1/20 0.36
MPO P05164 1/20 0.35
RORC P51449 1/20 0.35
STS P08842 1/20 0.35
HSD11B1 P28845 1/20 0.35
ESR2 Q92731 1/20 0.34
SPR P35270 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2885578 0.92 MEN1 (0.41) UCHL1HDAC1HDAC6NOTUMKDM1A
SCHEMBL2885604 0.90 UCHL1 (0.47) UCHL1HDAC1HDAC6NOTUMKDM1A
SCHEMBL3902861 0.82 UCHL1 (0.52) UCHL1HDAC1HDAC6NOTUMKDM1A
SCHEMBL31014046 0.82 UCHL1 (0.52) UCHL1HDAC1HDAC6NOTUMKDM1A
SCHEMBL30147617 0.78 UCHL1 (0.61) UCHL1HDAC1HDAC6NOTUMKDM1A
SCHEMBL20571008 0.78 UCHL1 (0.61) UCHL1HDAC1HDAC6NOTUMKDM1A
SCHEMBL868725 0.76 NOTUM (0.65) UCHL1HDAC1HDAC6NOTUMKDM1A
SCHEMBL20571049 0.76 UCHL1 (0.46) UCHL1HDAC1HDAC6NOTUMKDM1A
SCHEMBL3502782 0.75 UCHL1 (0.45) UCHL1HDAC1HDAC6NOTUMKDM1A
SCHEMBL2885921 0.75 NOTUM (0.47) UCHL1HDAC1HDAC6NOTUMKDM1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2121638-A2 NON-NUCLEOSIDE REVERSE TRANSCRIPTASE INHIBITORS Merck & Co., Inc. (US) 2009-11-25 EP disclosed
WO-2008076225-A2 NON-NUCLEOSIDE REVERSE TRANSCRIPTASE INHIBITORS MERCK & CO., INC. (US) 2008-06-26 WO disclosed