SCHEMBL4558593

SCHEMBL4558593

Cc1cc(Cl)cc2cc(C(=O)NC3CCCNC3)[nH]c12

nearest known ligand 0.51

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 5/20 0.51
SYK P43405 1/20 0.49
SMYD3 Q9H7B4 3/20 0.46
MAPK1 P28482 1/20 0.46
OPRK1 P41145 1/20 0.46
PBK Q96KB5 5/20 0.45
NSD2 O96028 1/20 0.43
SETD2 Q9BYW2 1/20 0.43
CDK2AP1 O14519 1/20 0.42
CHEK1 O14757 1/20 0.42
GHSR Q92847 2/20 0.41
CHRNA1 P02708 1/20 0.41
CHRNB2 P17787 1/20 0.41
CHRNB4 P30926 1/20 0.41
CHRNA4 P43681 1/20 0.41
TOP2A P11388 1/20 0.41
CYP1A2 P05177 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4558311 0.93 HRH4 (0.53) HRH4SYKSMYD3PBKNSD2
SCHEMBL3604185 0.89 SMYD3 (0.47) HRH4SYKSMYD3MAPK1OPRK1
SCHEMBL3604188 0.89 SMYD3 (0.47) HRH4SYKSMYD3MAPK1OPRK1
SCHEMBL25532114 0.84 MAPK1 (0.47) SYKSMYD3MAPK1OPRK1PBK
SCHEMBL3610802 0.83 SMYD3 (0.67) HRH4SYKSMYD3MAPK1OPRK1
SCHEMBL3610798 0.83 SMYD3 (0.67) HRH4SYKSMYD3MAPK1OPRK1
SCHEMBL3610639 0.81 SYK (0.51) SYKSMYD3MAPK1OPRK1PBK
SCHEMBL3610636 0.81 SYK (0.51) SYKSMYD3MAPK1OPRK1PBK
SCHEMBL3618497 0.81 SYK (0.51) SYKSMYD3MAPK1OPRK1PBK
SCHEMBL21225379 0.80 SYK (0.49) SYKMAPK1OPRK1PBKCDK2AP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009158375-A1 AZA-CYLIC INDOLE- 2 -CARBOXAMIDES AND METHODS OF USE THEREOF ABBOTT LABORATORIES (US) 2009-12-30 WO claimed