SCHEMBL4558788

SCHEMBL4558788

COCC(C(=O)O)c1ccc(-n2ccnn2)cc1

nearest known ligand 0.52

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 7/20 0.52
CYP19A1 P11511 4/20 0.47
MAPK1 P28482 1/20 0.42
CYP1A1 P04798 1/20 0.38
ALDH1A1 P00352 1/20 0.35
ELOVL1 Q9BW60 1/20 0.35
GLS O94925 1/20 0.35
MAPT P10636 1/20 0.34
CCKAR P32238 2/20 0.34
KDM4E B2RXH2 1/20 0.34
GAA P10253 1/20 0.34
HTT P42858 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4484833 0.85 NOTUM (0.56) NOTUMCYP19A1CYP1A1ELOVL1HTT
SCHEMBL17984479 0.83 NOTUM (0.48) NOTUMCYP19A1MAPK1CYP1A1ALDH1A1
SCHEMBL2387626 0.80 NOTUM (0.56) NOTUMCYP19A1MAPK1ALDH1A1
SCHEMBL9756479 0.77 NOTUM (0.66) NOTUMCYP19A1ALDH1A1ELOVL1GAA
SCHEMBL29211037 0.72 ESR1 (0.51) ALDH1A1MAPTGAAHTT
SCHEMBL2016945 0.71 CYP2C19 (0.52) MAPK1ALDH1A1GLS
SCHEMBL7336731 0.71 NOTUM (0.46) NOTUMCYP19A1MAPK1
SCHEMBL25201694 0.70 L3MBTL1 (0.42) ALDH1A1MAPTGAAHTT
SCHEMBL30387958 0.70 L3MBTL1 (0.42) ALDH1A1MAPTGAAHTT
SCHEMBL27751247 0.70 AKR1C3 (0.54) MAPTGAAHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2035396-A2 TRIAZOLE COMPOUNDS THAT MODULATE HSP90 ACTIVITY Synta Pharmaceuticals Corporation (US) 2009-03-18 EP claimed
WO-2007139967-A2 TRIAZOLE COMPOUNDS THAT MODULATE HSP90 ACTIVITY SYNTA PHARMACEUTICALS CORP. (US) 2007-12-06 WO claimed