SCHEMBL4559009

SCHEMBL4559009

c1cnnc(-n2ccnn2)c1

nearest known ligand 0.42

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 15/20 0.42
KEAP1 Q14145 1/20 0.42
MAP3K5 Q99683 1/20 0.41
CYP19A1 P11511 1/20 0.34
GOT1 P17174 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2C9 P11712 1/20 0.33
CHRNB2 P17787 1/20 0.33
CYP2B6 P20813 1/20 0.33
MAOA P21397 1/20 0.33
CYP2C19 P33261 1/20 0.33
CHRNA4 P43681 1/20 0.33
HTR3A P46098 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30643761 1.00 NOTUM (0.42) NOTUMKEAP1MAP3K5CYP19A1GOT1
SCHEMBL24240280 0.82 NOTUM (0.48) NOTUMKEAP1MAP3K5CYP19A1CYP1A2
SCHEMBL2086500 0.75 NOTUM (0.42) NOTUMKEAP1MAP3K5CYP19A1CYP1A2
SCHEMBL6482737 0.75 ALDH1A1 (0.48) NOTUMGOT1
SCHEMBL31359354 0.75 SMN1; SMN2 (0.46) NOTUMKEAP1MAP3K5
SCHEMBL503233 0.75 SMN1; SMN2 (0.46) NOTUMKEAP1MAP3K5
SCHEMBL17714528 0.73 NOTUM (0.48) NOTUM
SCHEMBL30948251 0.72 NOTUM (0.48) NOTUMKEAP1MAP3K5CYP19A1
SCHEMBL3148048 0.71 GOT1 (0.37) GOT1CYP1A2
SCHEMBL17104832 0.71 GOT1 (0.37) GOT1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009054789-A1 1,2,3-TRIAZOLE PYRROLIDINE DERIVATIVES AS MODULATORS OF MGLUR5 ASTRAZENECA AB (SE) 2009-04-30 WO claimed