SCHEMBL4559448

SCHEMBL4559448

Cc1nc(C(=O)N(C)CCN(C)c2nc3ccccc3o2)c(-c2ccccc2)s1

nearest known ligand 0.46

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 10/20 0.46
HCRTR2 O43614 7/20 0.46
PPARG P37231 8/20 0.43
PPARA Q07869 1/20 0.41
HDAC6 Q9UBN7 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4560777 0.89 HCRTR1 (0.54) HCRTR1HCRTR2PPARGPPARA
SCHEMBL4560318 0.87 HCRTR1 (0.49) HCRTR1HCRTR2PPARG
SCHEMBL4561212 0.82 HCRTR1 (0.53) HCRTR1HCRTR2PPARGPPARA
SCHEMBL3645277 0.77 HCRTR1 (0.50) HCRTR1HCRTR2
SCHEMBL2500909 0.75 HCRTR1 (0.54) HCRTR1HCRTR2
SCHEMBL2501264 0.75 HCRTR1 (0.54) HCRTR1HCRTR2
SCHEMBL3645275 0.72 PIN1 (0.58) HCRTR1HCRTR2
SCHEMBL2541745 0.72 PPARG (0.57) HCRTR1HCRTR2PPARGPPARAHDAC6
SCHEMBL13471010 0.70 PPARG (0.57) HCRTR1HCRTR2PPARGPPARAHDAC6
SCHEMBL2545232 0.69 HCRTR1 (0.59) HCRTR1HCRTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009011775-A1 AMIDOETHYL ALKYLAMINO OREXIN RECEPTOR ANTAGONISTS MERCK & CO., INC. (US) 2009-01-22 WO claimed
WO-2009011775-A1 AMIDOETHYL ALKYLAMINO OREXIN RECEPTOR ANTAGONISTS MERCK & CO., INC. (US) 2009-01-22 WO disclosed