SCHEMBL4560751

SCHEMBL4560751

COC(=O)c1sc(Nc2cc(OCc3ccc(OC)cc3)ccc2[N+](=O)[O-])cc1OC(C)c1ccccc1C(F)(F)F

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLK1 P53350 6/20 0.41
PLK3 Q9H4B4 3/20 0.41
AKR1B10 O60218 1/20 0.38
AKR1B1 P15121 1/20 0.38
AKR1C4 P17516 1/20 0.38
AKR1C3 P42330 1/20 0.38
AKR1C2 P52895 1/20 0.38
AKR1C1 Q04828 1/20 0.38
TP53 P04637 1/20 0.37
RXFP1 Q9HBX9 1/20 0.37
RAB9A P51151 2/20 0.36
AR P10275 2/20 0.36
PIK3CD O00329 1/20 0.36
PIK3C2B O00750 1/20 0.36
RIOK3 O14730 1/20 0.36
DAPK3 O43293 1/20 0.36
PIP5K1C O60331 1/20 0.36
RPS6KA4 O75676 1/20 0.36
STK10 O94804 1/20 0.36
PRKD3 O94806 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2982288 1.00 PLK1 (0.41) PLK1PLK3AKR1B10AKR1B1AKR1C4
SCHEMBL14568212 0.96 PLK1 (0.39) PLK1PLK3AKR1B10AKR1B1AKR1C4
SCHEMBL13592940 0.96 PLK1 (0.39) PLK1PLK3AKR1B10AKR1B1AKR1C4
SCHEMBL2973849 0.94 AKR1C3 (0.41) PLK1PLK3AKR1B10AKR1B1AKR1C4
SCHEMBL2973853 0.94 AKR1C3 (0.41) PLK1PLK3AKR1B10AKR1B1AKR1C4
SCHEMBL2986971 0.91 PLK1 (0.41) PLK1PLK3AKR1B10AKR1B1AKR1C4
SCHEMBL5582470 0.89 AKR1B10 (0.39) PLK1PLK3AKR1B10AKR1B1AKR1C4
SCHEMBL2982204 0.89 AKR1B10 (0.39) PLK1PLK3AKR1B10AKR1B1AKR1C4
SCHEMBL13592925 0.89 AKR1B10 (0.39) AKR1B10AKR1B1AKR1C4AKR1C3AKR1C2
SCHEMBL2987859 0.88 PLK1 (0.44) PLK1PLK3TP53RXFP1AR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1924572-B1 REGIOSELECTIVE PROCESS FOR PREPARING BENZIMIDAZOLE THIOPHENES SMITHKLINE BEECHAM CORP (US) 2009-12-30 EP disclosed