SCHEMBL456089

SCHEMBL456089

[CH2]CCCc1nc(-c2cccc(N)c2)c[nH]1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.42
KDM4E B2RXH2 4/20 0.42
MEN1 O00255 4/20 0.42
MAPT P10636 3/20 0.42
HPGD P15428 3/20 0.42
KMT2A Q03164 3/20 0.42
LMNA P02545 3/20 0.42
METAP2 P50579 1/20 0.41
NPC1 O15118 3/20 0.39
RAB9A P51151 3/20 0.39
TSHR P16473 1/20 0.39
RECQL P46063 1/20 0.39
GLA P06280 1/20 0.39
KDM1A O60341 1/20 0.38
MAOA P21397 1/20 0.36
TP53 P04637 2/20 0.35
NFKB1 P19838 1/20 0.35
NFKB2 Q00653 1/20 0.35
RELA Q04206 1/20 0.35
ATAD2 Q6PL18 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5673498 0.83 SMN1; SMN2 (0.36) ALDH1A1MEN1HPGDKMT2ARAB9A
SCHEMBL455756 0.77 MAPK1 (0.42) ALDH1A1METAP2AXLMKNK1MKNK2
SCHEMBL453941 0.77
SCHEMBL4861987 0.76 GSK3B (0.43) MAPTLMNANPC1RAB9A
SCHEMBL4703629 0.75 HPGD (0.38) ALDH1A1KDM4EMEN1MAPTHPGD
SCHEMBL5500501 0.73 SMN1; SMN2 (0.38) ALDH1A1MEN1HPGDKMT2ARAB9A
SCHEMBL4704287 0.72 MAPT (0.43) ALDH1A1KDM4EMEN1MAPTHPGD
SCHEMBL11097956 0.71 SSTR1 (0.43) ALDH1A1MEN1KMT2ARAB9AMAOA
SCHEMBL7056243 0.70 TSHR (0.54) ALDH1A1KDM4EMEN1MAPTHPGD
SCHEMBL5004823 0.70 ALDH1A1 (0.50) ALDH1A1KDM4EMEN1MAPTHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2613630-A1 HYDROGEN BOND FORMING FLUORO KETOLIDES FOR TREATING DISEASES Cempra Pharmaceuticals, Inc. (US) 2013-07-17 EP disclosed
WO-2012034058-A1 HYDROGEN BOND FORMING FLUORO KETOLIDES FOR TREATING DISEASES CEMPRA PHARMACEUTICALS, INC. (US) 2012-03-15 WO disclosed