SCHEMBL4562797

SCHEMBL4562797

O=C(NO)c1cnc(N2CCNCC2)nc1-c1ccccc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 13/20 0.51
HIF1A Q16665 12/20 0.51
CYP1A2 P05177 12/20 0.51
CASP1 P29466 11/20 0.51
CASP7 P55210 11/20 0.51
HSD17B10 Q99714 10/20 0.51
HPGD P15428 9/20 0.51
CYP2C9 P11712 7/20 0.51
CYP2C19 P33261 5/20 0.51
GLA P06280 3/20 0.51
CYP3A4 P08684 10/20 0.50
USP2 O75604 9/20 0.50
ALOX15 P16050 1/20 0.50
LMNA P02545 4/20 0.45
PTPN11 Q06124 4/20 0.45
KMT2A Q03164 2/20 0.45
KDM4E B2RXH2 1/20 0.45
S1PR2 O95136 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
TP53 P04637 4/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6016398 0.88 ALDH1A1 (0.55) ALDH1A1HIF1ACYP1A2CASP1CASP7
SCHEMBL12485766 0.82 ALDH1A1 (0.47) ALDH1A1HIF1ACYP1A2CASP1CASP7
SCHEMBL973782 0.80 MMP2 (0.51) CYP2C9CYP2C19TSHR
SCHEMBL4562795 0.79 CYP1A2 (0.44) ALDH1A1CYP1A2CYP2C19CYP3A4ALOX15
SCHEMBL4112334 0.77 ALDH1A1 (0.54) ALDH1A1HIF1ACYP1A2CASP1CASP7
Piperazine SCHEMBL6016590 0.76 ALDH1A1 (0.53) ALDH1A1HIF1ACYP1A2CASP1CASP7
SCHEMBL4124274 0.75 ALDH1A1 (0.43) ALDH1A1HIF1ACYP1A2CASP1CASP7
SCHEMBL6016426 0.75 PTPN11 (0.53) ALDH1A1CASP1CASP7HSD17B10HPGD
SCHEMBL976971 0.74 MEN1 (0.74) ALDH1A1CYP1A2HPGDCYP2C9CYP2C19
Hydrochloric Acid SCHEMBL3866277 0.74 PTPN11 (0.52) ALDH1A1CASP1CASP7HSD17B10HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009114470-A2 TETRAHYDROINDOLE AND TETRAHDYROINDAZOLE AS HSP90 INHIBITORS CONTAINING A ZINC BINDING MOIETY CURIS, INC. (US) 2009-09-17 WO disclosed