SCHEMBL4563231

SCHEMBL4563231

COCCOC(=O)Oc1cn(C)nc1C(F)F

nearest known ligand 0.32

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.32
GAA P10253 1/20 0.32
IRAK4 Q9NWZ3 1/20 0.31
TP53 P04637 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4563987 0.87 TSHR (0.32) TSHRTP53
SCHEMBL1012200 0.85 ADORA2A (0.36) GAATP53
SCHEMBL1396811 0.84 KDM4E (0.36) GAAIRAK4
SCHEMBL2248952 0.80 TSHR (0.47) TSHRGAAIRAK4TP53
SCHEMBL3118115 0.78 ALDH1A1 (0.34) TSHR
SCHEMBL27774048 0.77 HIF1A (0.37) GAAIRAK4
SCHEMBL1136291 0.77 GAA (0.31) GAAIRAK4
SCHEMBL27753360 0.77 CYP4F2 (0.34) TSHRGAAIRAK4
SCHEMBL2576002 0.76 IRAK4 (0.33) GAAIRAK4
SCHEMBL1135830 0.76 IRAK4 (0.33) GAAIRAK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2121618-A1 PROCESS FOR PREPARING FLUOROMETHYL-SUBSTITUTED HETEROCYCLIC COMPOUNDS BASF SE (DE) 2009-11-25 EP disclosed
WO-2008077907-A1 PROCESS FOR PREPARING FLUOROMETHYL-SUBSTITUTED HETEROCYCLIC COMPOUNDS BASF SE (DE) 2008-07-03 WO disclosed