SCHEMBL4564958

SCHEMBL4564958

c1ccc(C[C@H]2c3ccc(OC4CCNCC4)cc3CC23CCNCC3)cc1

nearest known ligand 0.50

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HRH1 P35367 5/20 0.50
DYRK1A Q13627 1/20 0.39
GBA1 P04062 1/20 0.39
HRH3 Q9Y5N1 2/20 0.38
KHK P50053 2/20 0.38
SLC6A2 P23975 3/20 0.36
SLC6A3 Q01959 3/20 0.36
HTR1A P08908 2/20 0.36
HTR6 P50406 1/20 0.36
IKBKB O14920 1/20 0.36
NMT1 P30419 1/20 0.36
HTR2A P28223 1/20 0.35
HTR2C P28335 1/20 0.35
SLC6A4 P31645 1/20 0.35
HTR7 P34969 1/20 0.35
HTR2B P41595 1/20 0.35
HTR3A P46098 1/20 0.35
HTR4 Q13639 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4478245 0.87 HRH3 (0.48) HRH1HRH3
SCHEMBL4481591 0.87 HRH1 (0.42) HRH1HTR2C
SCHEMBL4484620 0.85 HTR2A (0.41) HRH1SLC6A2SLC6A3HTR1AHTR2A
SCHEMBL3799816 0.70 TSHR (0.52) HRH1HRH3
SCHEMBL19023362 0.68 HRH1 (0.56) HRH1HRH3KHKSLC6A2SLC6A3
SCHEMBL24437475 0.68 HRH1 (1.00) HRH1GBA1KHKSLC6A2SLC6A3
SCHEMBL12420648 0.68 HRH1 (0.82) HRH1GBA1HRH3KHKSLC6A2
SCHEMBL12735765 0.68 HRH1 (0.61) HRH1SLC6A2SLC6A3HTR1AHTR2C
Hydrochloric Acid SCHEMBL2195506 0.67 HRH1 (0.59) HRH1SLC6A2SLC6A3HTR1AHTR2C
SCHEMBL4335524 0.67 AR (0.40) HRH1SLC6A2SLC6A3HTR1AHTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009039431-A2 SUBSTITUTED ARYL-FUSED SPIROCYCLIC AMINES NEUROGEN CORPORATION (US) 2009-03-26 WO disclosed