SCHEMBL4484620

SCHEMBL4484620

COc1ccc2c(c1)CC1(CCNCC1)[C@H]2Cc1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 1/20 0.41
TACR1 P25103 1/20 0.40
HTR2C P28335 2/20 0.40
EED O75530 1/20 0.39
SLC6A2 P23975 2/20 0.39
SLC6A4 P31645 1/20 0.39
NPY5R Q15761 1/20 0.39
CHRNB2 P17787 1/20 0.38
CHRNB4 P30926 1/20 0.38
CHRNA3 P32297 1/20 0.38
CHRNA7 P36544 1/20 0.38
CHRNA4 P43681 1/20 0.38
SIGMAR1 Q99720 3/20 0.38
HTR1A P08908 2/20 0.38
AR P10275 2/20 0.37
GRIN1 Q05586 1/20 0.37
GRIN2B Q13224 1/20 0.37
ADRB2 P07550 1/20 0.37
ADRA2A P08913 1/20 0.37
ADRA2B P18089 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4564958 0.85 HRH1 (0.50) HTR2AHTR2CSLC6A2SLC6A4HTR1A
SCHEMBL4335524 0.80 AR (0.40) HTR2AHTR2CSLC6A2SIGMAR1HTR1A
SCHEMBL4478245 0.78 HRH3 (0.48) HRH1
SCHEMBL4481591 0.78 HRH1 (0.42) HTR2CHRH1OPRK1
SCHEMBL23508701 0.77 HTR2C (0.45) HTR2AHTR2CSLC6A2CHRNB2CHRNB4
SCHEMBL25707304 0.77 HTR2C (0.45) HTR2AHTR2CSLC6A2CHRNB2CHRNB4
Hydrochloric Acid SCHEMBL30486474 0.76 HTR2C (0.44) HTR2AHTR2CSLC6A2CHRNB2CHRNB4
Hydrochloric Acid SCHEMBL30486634 0.76 HTR2C (0.44) HTR2AHTR2CSLC6A2CHRNB2CHRNB4
Hydrochloric Acid SCHEMBL25347445 0.76 HTR2C (0.44) HTR2AHTR2CSLC6A2CHRNB2CHRNB4
SCHEMBL24879518 0.75 HTR2C (0.56) HTR2AHTR2CSLC6A2SIGMAR1HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009039431-A2 SUBSTITUTED ARYL-FUSED SPIROCYCLIC AMINES NEUROGEN CORPORATION (US) 2009-03-26 WO disclosed