SCHEMBL4565202

SCHEMBL4565202

CC(C)(C)N(C(=O)O)[C@@H]1CCCN(C(=O)C(c2cccc(OC(F)(F)F)c2)C2CCCCC2)C1

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CHRM3 P20309 4/20 0.41
NOTUM Q6P988 1/20 0.39
EPHX1 P07099 1/20 0.37
CCR5 P51681 2/20 0.37
BCL9 O00512 1/20 0.37
CTNNB1 P35222 1/20 0.37
UBE2M P61081 1/20 0.37
DCUN1D1 Q96GG9 1/20 0.37
USP30 Q70CQ3 1/20 0.37
SLC6A2 P23975 5/20 0.36
FFAR1 O14842 3/20 0.36
PPARA Q07869 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4565133 0.90 CHRM3 (0.45) CHRM3NOTUMEPHX1CCR5UBE2M
SCHEMBL4512194 0.85 SLC6A2 (0.45) NOTUMBCL9CTNNB1UBE2MDCUN1D1
SCHEMBL4510883 0.85 SLC6A2 (0.45) NOTUMBCL9CTNNB1UBE2MDCUN1D1
SCHEMBL4117389 0.81 CHRM3 (0.42) CHRM3NOTUMEPHX1USP30
SCHEMBL4847784 0.81 CHRM3 (0.42) CHRM3NOTUMEPHX1USP30
SCHEMBL4493804 0.81 SLC6A2 (0.45) NOTUMUBE2MDCUN1D1SLC6A2
SCHEMBL4497752 0.81 SLC6A2 (0.45) NOTUMUBE2MDCUN1D1SLC6A2
SCHEMBL4847465 0.78 CHRM3 (0.43) CHRM3NOTUMEPHX1
SCHEMBL4955085 0.78 CHRM3 (0.43) CHRM3NOTUMEPHX1
SCHEMBL4503886 0.75 SLC6A2 (0.47) UBE2MDCUN1D1SLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7491723-B2 Alkanol and cycloalkanol-amine derivatives and methods of their use WYETH (US) 2009-02-17 US disclosed