SCHEMBL4565224

SCHEMBL4565224

Nc1ccc2c(C[O])n[nH]c2n1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 5/20 0.42
ADORA2A P29274 4/20 0.42
CA5A P35218 1/20 0.39
MAPK13 O15264 2/20 0.33
MAPK12 P53778 2/20 0.33
MAPK11 Q15759 2/20 0.33
MAPK14 Q16539 2/20 0.33
PRMT5 O14744 1/20 0.32
GABRP O00591 2/20 0.31
GABRD O14764 2/20 0.31
GABRA1 P14867 2/20 0.31
GABRB1 P18505 2/20 0.31
GABRG2 P18507 2/20 0.31
GABRB3 P28472 2/20 0.31
GABRA5 P31644 2/20 0.31
GABRA3 P34903 2/20 0.31
GABRA2 P47869 2/20 0.31
GABRB2 P47870 2/20 0.31
GABRA4 P48169 2/20 0.31
GABRE P78334 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31207340 0.77 ADORA1 (0.46) ADORA1ADORA2ACA5AMAPK13MAPK12
SCHEMBL25475233 0.72 ADORA1 (0.50) ADORA1ADORA2ACA5AMAPK13MAPK12
SCHEMBL32683505 0.72 ADORA1 (0.50) ADORA1ADORA2ACA5AMAPK13MAPK12
SCHEMBL493663 0.70 ADORA1 (0.41) ADORA1ADORA2ACA5AGABRPGABRD
SCHEMBL30554311 0.67 MAPK13 (0.47) ADORA1ADORA2ACA5AMAPK13MAPK12
SCHEMBL20916782 0.67 MAPK13 (0.47) ADORA1ADORA2ACA5AMAPK13MAPK12
SCHEMBL29768213 0.62 PDPK1 (0.46) ADORA1ADORA2APDPK1
SCHEMBL26675355 0.62 PDPK1 (0.46) ADORA1ADORA2APDPK1
SCHEMBL7425108 0.59 PDPK1 (0.35) PDPK1
SCHEMBL31032821 0.58 CCR1 (0.41) PDPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009117278-A2 PROCESSES FOR PREPARING (AMINO-PYRAZOLOPYRIDINYL)METHOXY SUBSTITUTED BIARYL ETHERS MERCK & CO., INC. (US) 2009-09-24 WO disclosed