SCHEMBL4565646

SCHEMBL4565646

Cc1cnc(Cc2cnc(CC(N)CCCN(C)C(=O)Nc3ncc[nH]3)c3ccccc23)c(C)c1

nearest known ligand 0.33

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CCKBR P32239 1/20 0.33
PTGES O14684 4/20 0.31
CXCR4 P61073 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4205917 0.74 PTGES (0.36) PTGES
SCHEMBL2084500 0.73 CXCR4 (0.36) PTGESCXCR4
SCHEMBL2084498 0.73
SCHEMBL4538831 0.68 ADORA2A (0.31) CXCR4
SCHEMBL4565645 0.68 MAPK1 (0.35) PTGES
SCHEMBL2085313 0.63 MAPK1 (0.39) PTGESCXCR4
SCHEMBL23428823 0.61 CXCR4 (0.30) CXCR4
SCHEMBL2085676 0.60 CXCR4 (0.38) CXCR4
SCHEMBL4206736 0.59 CXCR4 (0.42) CXCR4
Ammonia Solution, Strong SCHEMBL5574435 0.58 CXCR4 (0.50) CXCR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1613613-A4 CXCR4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC (CA) 2009-03-25 EP disclosed
EP-1613613-A2 CXCR4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2006-01-11 EP disclosed
WO-2004091518-A2 CXCR4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2004-10-28 WO disclosed