SCHEMBL4565645

SCHEMBL4565645

Cc1cnc(CC(CCCNCc2nccc3ccccc23)N(C)C(=O)Nc2ncc[nH]2)c(C)c1

nearest known ligand 0.35

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 1/20 0.35
SLC40A1 Q9NP59 1/20 0.32
PTGES O14684 2/20 0.31
F2 P00734 1/20 0.30
F10 P00742 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2084500 0.76 CXCR4 (0.36) MAPK1PTGES
SCHEMBL2084498 0.76
SCHEMBL5576013 0.74 CYP2A6 (0.38) MAPK1SLC40A1F2F10
SCHEMBL2085313 0.72 MAPK1 (0.39) MAPK1SLC40A1PTGES
SCHEMBL4205917 0.71 PTGES (0.36) MAPK1SLC40A1PTGES
SCHEMBL5576002 0.70 CXCR4 (0.37) SLC40A1
SCHEMBL4565646 0.68 CCKBR (0.33) PTGES
SCHEMBL2083396 0.68 JUN (0.37) MAPK1
SCHEMBL2080968 0.65 CXCR4 (0.39) MAPK1F2F10
SCHEMBL2085676 0.65 CXCR4 (0.38) MAPK1F2F10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1613613-A4 CXCR4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC (CA) 2009-03-25 EP disclosed
EP-1613613-A2 CXCR4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2006-01-11 EP disclosed
WO-2004091518-A2 CXCR4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2004-10-28 WO disclosed