SCHEMBL4565678

SCHEMBL4565678

COc1cccc2c1OCC1C2N(Br)c2ccc(C(N)=S)cc2C1(C)C

nearest known ligand 0.39

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ACHE P22303 3/20 0.33
BCHE P06276 2/20 0.33
KDM4E B2RXH2 1/20 0.32
SMN1; SMN2 Q16637 2/20 0.31
LMNA P02545 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2D6 P10635 1/20 0.31
CYP2C19 P33261 1/20 0.31
ALDH1A1 P00352 2/20 0.31
HPGD P15428 1/20 0.31
TERT O14746 1/20 0.31
PKM P14618 1/20 0.30
BACE1 P56817 1/20 0.30
MAPK1 P28482 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4563417 0.92 ACHE (0.36) ACHEBCHEKDM4ESMN1; SMN2LMNA
SCHEMBL4629041 0.83 ACHE (0.34) ACHEBCHEKDM4ESMN1; SMN2LMNA
SCHEMBL4563342 0.81 PSMB5 (0.34) ACHEBCHEKDM4ESMN1; SMN2LMNA
SCHEMBL4627058 0.80 KDM4E (0.34) ACHEBCHEKDM4ESMN1; SMN2LMNA
SCHEMBL4564292 0.78 F2 (0.34) KDM4ESMN1; SMN2LMNACYP3A4CYP2D6
SCHEMBL4626708 0.78 MEN1 (0.35) KDM4ETERT
SCHEMBL4884510 0.73 F2 (0.32) ALDH1A1
SCHEMBL4554178 0.70 IRAK4 (0.35) KDM4ESMN1; SMN2LMNACYP3A4CYP2D6
SCHEMBL4884506 0.67 ALDH1A1 (0.33) SMN1; SMN2LMNAALDH1A1HPGDPKM
SCHEMBL4555663 0.67 MAPT (0.38) KDM4ESMN1; SMN2ALDH1A1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2125825-A1 ABCA1 ELEVATING COMPOUNDS CV THERAPEUTICS, INC. (US) 2009-12-02 EP disclosed
WO-2008079139-A1 ABCA1 ELEVATING COMPOUNDS CV THERAPEUTICS, INC. (US) 2008-07-03 WO disclosed
EP-1907395-A1 ABCA1 ELEVATING COMPOUNDS CV THERAPEUTICS, INC. (US) 2008-04-09 EP disclosed
WO-2007002867-A1 ABCA1 ELEVATING COMPOUNDS CV THERAPEUTICS, INC. (US) 2007-01-04 WO disclosed