SCHEMBL4565949

SCHEMBL4565949

CNc1ccc(-c2cc3cc(F)ccc3n2C(=O)O)cn1

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TDO2 P48775 3/20 0.44
FYN P06241 1/20 0.41
MKNK1 Q9BUB5 1/20 0.41
HCAR3 P49019 1/20 0.40
HPGD P15428 2/20 0.39
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
HSD17B10 Q99714 1/20 0.39
SCD O00767 1/20 0.39
NR1H2 P55055 1/20 0.38
ABL1 P00519 2/20 0.38
NTRK1 P04629 1/20 0.38
APP P05067 5/20 0.37
MAPT P10636 1/20 0.36
NNMT P40261 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3305065 0.85 NR1H2 (0.53) NR1H2
SCHEMBL3309831 0.80 GRM2 (0.38) HPGDKDM4EALDH1A1HSD17B10NR1H2
SCHEMBL27830572 0.77 ACLY (0.47) TDO2NTRK1MAPT
SCHEMBL3301415 0.72 NR1H2 (0.53) NR1H2APP
SCHEMBL31196173 0.71 AOC3 (0.47) HPGDALDH1A1HSD17B10ABL1
SCHEMBL17674258 0.70 KDM4E (0.46) HPGDKDM4EALDH1A1HSD17B10ABL1
SCHEMBL17674201 0.69 NTRK1 (0.48) HPGDKDM4EALDH1A1HSD17B10NTRK1
SCHEMBL4054875 0.69 KDM4E (0.53) HPGDKDM4EALDH1A1HSD17B10
SCHEMBL17674413 0.68 KDM4E (0.43) HPGDKDM4EALDH1A1HSD17B10NTRK1
SCHEMBL4437497 0.67 NR1H2 (0.51) NR1H2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2121655-A1 NOVEL 2-HETEROARYL SUBSTITUTED INDOLES 695 AstraZeneca AB (SE) 2009-11-25 EP disclosed
WO-2008108729-A1 NOVEL 2-HETEROARYL SUBSTITUTED INDOLES 695 ASTRAZENECA AB (SE) 2008-09-12 WO disclosed