SCHEMBL4566517

SCHEMBL4566517

O=C(O)c1ccc(N2CCN(c3ccc(-c4nc5cc(C(F)(F)F)ccc5[nH]4)cn3)CC2)nc1

nearest known ligand 0.60

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 19/20 0.60
KCNH2 Q12809 11/20 0.60
SOAT1 P35610 3/20 0.59
ADORA2A P29274 2/20 0.59
CYP2C9 P11712 2/20 0.57
CYP3A4 P08684 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10082142 0.86 DGAT1 (0.55) DGAT1KCNH2SOAT1ADORA2ACYP2C9
SCHEMBL4561861 0.85 DGAT1 (0.65) DGAT1KCNH2SOAT1ADORA2ACYP2C9
SCHEMBL4560992 0.85 DGAT1 (0.57) DGAT1KCNH2SOAT1ADORA2ACYP2C9
SCHEMBL4560514 0.84 DGAT1 (0.62) DGAT1KCNH2SOAT1ADORA2ACYP2C9
SCHEMBL10147125 0.84 DGAT1 (0.58) DGAT1KCNH2CYP2C9CYP3A4
SCHEMBL14235399 0.83 DGAT1 (0.60) DGAT1KCNH2SOAT1ADORA2ACYP2C9
SCHEMBL14128713 0.83 DGAT1 (0.60) DGAT1KCNH2SOAT1ADORA2ACYP2C9
SCHEMBL10147139 0.83 ACACB (0.57) DGAT1KCNH2CYP2C9CYP3A4
SCHEMBL6995535 0.83 DGAT1 (0.61) DGAT1KCNH2SOAT1ADORA2ACYP2C9
SCHEMBL10147228 0.82 DGAT1 (0.89) DGAT1KCNH2CYP2C9CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012064569-A1 IMIDAZOLE DERIVATIVES MERCK SHARP & DOHME CORP. (US) 2012-05-18 WO disclosed