SCHEMBL6995535

SCHEMBL6995535

FC(F)(F)c1ccc2[nH]c(-c3ccc(N4CCCN(c5ccccc5)CC4)nc3)nc2c1

nearest known ligand 0.61

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 19/20 0.61
KCNH2 Q12809 5/20 0.59
SOAT1 P35610 3/20 0.59
ADORA2A P29274 1/20 0.52
CYP3A4 P08684 1/20 0.51
CYP2C9 P11712 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4561861 0.97 DGAT1 (0.65) DGAT1KCNH2SOAT1ADORA2ACYP3A4
SCHEMBL4566817 0.85 DGAT1 (0.60) DGAT1KCNH2SOAT1ADORA2ACYP3A4
SCHEMBL4560514 0.84 DGAT1 (0.62) DGAT1KCNH2SOAT1ADORA2ACYP3A4
SCHEMBL4562655 0.83 DGAT1 (0.62) DGAT1KCNH2SOAT1ADORA2ACYP3A4
SCHEMBL4566517 0.83 DGAT1 (0.60) DGAT1KCNH2SOAT1ADORA2ACYP3A4
SCHEMBL6994712 0.82 DGAT1 (0.54) DGAT1KCNH2ADORA2ACYP2C9
SCHEMBL19175769 0.81 DGAT1 (0.77) DGAT1KCNH2SOAT1ADORA2ACYP3A4
SCHEMBL19137929 0.80 DGAT1 (0.64) DGAT1KCNH2SOAT1
SCHEMBL10326124 0.80 DGAT1 (0.68) DGAT1KCNH2SOAT1ADORA2ACYP3A4
SCHEMBL10146471 0.78 DGAT1 (0.60) DGAT1KCNH2SOAT1CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012064569-A1 IMIDAZOLE DERIVATIVES MERCK SHARP & DOHME CORP. (US) 2012-05-18 WO disclosed