SCHEMBL4566535

SCHEMBL4566535

O=C(O)c1cc2cc(Cl)ccc2n1CCN1CCOCC1

nearest known ligand 0.57

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CCR2 P41597 13/20 0.57
MAPT P10636 2/20 0.48
TP53 P04637 1/20 0.48
MAPK1 P28482 1/20 0.48
HTT P42858 1/20 0.48
ATM Q13315 1/20 0.48
PTGS2 P35354 1/20 0.47
ALDH1A1 P00352 1/20 0.47
KMT2A Q03164 1/20 0.47
CNR2 P34972 1/20 0.47
ABCB11 O95342 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6752517 0.90 CCR2 (0.56) CCR2MAPTTP53MAPK1HTT
SCHEMBL6753789 0.84 CCR2 (0.53) CCR2MAPTTP53ALDH1A1KMT2A
SCHEMBL6753297 0.83 ALDH1A1 (0.56) CCR2MAPTALDH1A1KMT2ACNR2
SCHEMBL30121932 0.83 ALDH1A1 (0.56) CCR2MAPTALDH1A1KMT2ACNR2
SCHEMBL4539709 0.82 ALDH1A1 (0.57) CCR2MAPTTP53MAPK1ALDH1A1
SCHEMBL670091 0.79 MAPT (0.52) MAPTTP53MAPK1HTTATM
SCHEMBL8687383 0.79 CCR2 (0.62) CCR2ABCB11
SCHEMBL6750687 0.78 ALDH1A1 (0.53) CCR2ALDH1A1CNR2
SCHEMBL6754276 0.78 CCR9 (0.54) CCR2TP53
SCHEMBL16235858 0.76 CCR2 (0.59) CCR2ABCB11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009063495-A2 SUBSTITUTED INDOLE AND ITS DERIVATIVES AS CANNABINOID MODULATORS CADILA HEALTHCARE LIMITED (IN) 2009-05-22 WO claimed
WO-2009063495-A2 SUBSTITUTED INDOLE AND ITS DERIVATIVES AS CANNABINOID MODULATORS CADILA HEALTHCARE LIMITED (IN) 2009-05-22 WO disclosed