SCHEMBL456745

SCHEMBL456745

CCCCCCCC/C=C\CCCCCCCC(=O)N(C(=O)CCCCCCC/C=C\CCCCCCCC)C(P)(CO)C(=O)O

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PPARG P37231 5/20 0.53
PPARD Q03181 5/20 0.53
PPARA Q07869 5/20 0.53
F7 P08709 4/20 0.53
F3 P13726 4/20 0.53
TERT O14746 3/20 0.53
PTPN1 P18031 3/20 0.53
HSD17B10 Q99714 3/20 0.53
FABP4 P15090 3/20 0.53
MAPT P10636 2/20 0.53
BLM P54132 2/20 0.53
LMNA P02545 2/20 0.53
ALOX15 P16050 2/20 0.53
DUSP3 P51452 2/20 0.53
CYP19A1 P11511 2/20 0.53
PTGS1 P23219 2/20 0.53
NR4A2 P43354 2/20 0.53
SIRT6 Q8N6T7 2/20 0.53
PTPN7 P35236 2/20 0.53
TDP1 Q9NUW8 2/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1271901 1.00 PPARG (0.53) PPARGPPARDPPARAF7F3
SCHEMBL1470099 1.00 PPARG (0.53) PPARGPPARDPPARAF7F3
SCHEMBL1273217 0.91 GPR84 (0.44) PPARGPPARDPPARAPTPN1HSD17B10
SCHEMBL5490197 0.91 GPR84 (0.44) PPARGPPARDPPARAPTPN1HSD17B10
SCHEMBL45203 0.91 GPR84 (0.44) PPARGPPARDPPARAPTPN1HSD17B10
SCHEMBL30413 0.91 GPR84 (0.44) PPARGPPARDPPARAPTPN1HSD17B10
SCHEMBL253962 0.91 GPR84 (0.44) PPARGPPARDPPARAPTPN1HSD17B10
SCHEMBL5495040 0.91 GPR84 (0.44) PPARGPPARDPPARAPTPN1HSD17B10
SCHEMBL5395520 0.89 AKR1B1 (0.42) PPARGPPARDPPARAPTPN1HSD17B10
SCHEMBL786356 0.84 EPHX2 (0.47) PPARGPPARDPPARAF7F3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 2062 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4398882-A1 LIPID-BASED RNA FORMULATIONS SUITABLE FOR THERAPY BioNTech SE (DE) 2024-07-17 EP claimed
US-20240226325-A1 CATIONIC LIPIDS AND COMPOSITIONS THEREOF GENERATION BIO CO. 2024-07-11 US claimed
EP-4382094-A1 ATHEROSCLEROSIS-TARGETED LIPOSOME NANOCARRIER DELIVERY SYSTEM AND PREPARATION METHOD THEREFOR Beijing Inno Medicine Co., Ltd. (CN) 2024-06-12 EP claimed
WO-2024119017-A1 SYNTHETIC SINGLE STRANDED NUCLEIC ACID COMPOSITIONS AND METHODS THEREOF GENERATION BIO CO. (US) 2024-06-06 WO claimed
US-20240180940-A1 MPLA COMPOSITIONS AND METHODS OF USE REVELATION BIOSCIENCES, INC. 2024-06-06 US claimed
WO-2024119074-A1 STEALTH LIPID NANOPARTICLE COMPOSITIONS FOR CELL TARGETING GENERATION BIO CO. (US) 2024-06-06 WO claimed
WO-2024109929-A1 IONIZABLE LIPID AND USE THEREOF 艾斯拓康医药科技(北京)有限公司 2024-05-30 WO claimed
US-20240173267-A1 COMPOUNDS, COMPOSITIONS, AND METHODS OF USING THEREOF ONCORUS, INC. (US) 2024-05-30 US claimed
EP-4370135-A2 SINGLE CHAIN VARIABLE FRAGMENT (SCFV) MODIFIED LIPID NANOPARTICLE COMPOSITIONS AND USES THEREOF Generation Bio Co. (US) 2024-05-22 EP claimed
WO-2024094027-A1 BLOCKING SEQUENCE, KIT THEREOF, AND METHOD FOR USING SAME 深圳鸿生生物科技有限公司 2024-05-10 WO claimed
WO-1999040789-A1 METHODS AND COMPOUNDS FOR THE GENETIC TREATMENT OF HYPERLIPIDEMIA REGENTS OF THE UNIVERSITY OF MINNESOTA (US) 1999-08-19 WO claimed
WO-1999030686-A1 CATIONIC DRUGS ENCAPSULATED IN ANIONIC LIPOSOMES INEX PHARMACEUTICALS CORP. (CA) 1999-06-24 WO claimed
US-5874075-A STABILITY; HEAT RESISTANCE; ANTIAGGREGATION; NONDENATURING AMGEN INC. (US) 1999-02-23 US claimed
JP-2852127-B2 1999-01-27 JP claimed
WO-1998049350-B1 IN VIVO USE OF RECOMBINAGENIC OLIGONUCLEOBASES TO CORRECT GENETIC LESIONS IN HEPATOCYTES 1999-01-07 WO claimed
WO-1998049350-A1 IN VIVO USE OF RECOMBINAGENIC OLIGONUCLEOBASES TO CORRECT GENETIC LESIONS IN HEPATOCYTES REGENTS OF THE UNIVERSITY OF MINNESOTA (US) 1998-11-05 WO claimed
EP-0817614-A1 STABLE PROTEIN:PHOSPHOLIPID COMPOSITIONS AND METHODS------------ AMGEN INC. (US) 1998-01-14 EP claimed
WO-1996029989-A1 STABLE PROTEIN:PHOSPHOLIPID COMPOSITIONS AND METHODS____________ AMGEN INC. (US) 1996-10-03 WO claimed
EP-0671905-A1 STABLE PROTEIN: PHOSPHOLIPID COMPOSITIONS AND METHODS AMGEN INC. (US) 1995-09-20 EP claimed
WO-1995009611-A2 STABLE PROTEIN: PHOSPHOLIPID COMPOSITIONS AND METHODS AMGEN INC. (US) 1995-04-13 WO claimed