SCHEMBL4569737

SCHEMBL4569737

CC(C)(C)CN(Cc1cc(Br)n(S(=O)(=O)c2cccc(F)c2)c1)C(=O)O

nearest known ligand 0.42

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PTGDR Q13258 2/20 0.42
PTGDR2 Q9Y5Y4 2/20 0.42
PKM P14618 1/20 0.38
TSHR P16473 1/20 0.38
HTR6 P50406 2/20 0.37
PTGER2 P43116 2/20 0.36
TAS2R14 Q9NYV8 2/20 0.36
CHRM5 P08912 3/20 0.36
RAB9A P51151 1/20 0.36
MEN1 O00255 1/20 0.36
ALDH1A1 P00352 1/20 0.36
LMNA P02545 1/20 0.36
KMT2A Q03164 1/20 0.36
TSPO P30536 1/20 0.35
LIMK2 P53671 1/20 0.35
HCRTR2 O43614 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1156624 0.90 CHRM5 (0.43) HTR6CHRM5MEN1LMNAKMT2A
SCHEMBL1156488 0.89 CHRM5 (0.36) PTGDR2CHRM5ALDH1A1KMT2A
SCHEMBL1156885 0.89 PTGDR2 (0.40) PTGDRPTGDR2PKMHTR6TAS2R14
SCHEMBL1156564 0.88 LMNA (0.41) PTGDR2HTR6PTGER2CHRM5MEN1
SCHEMBL4411754 0.88 CHRM5 (0.42) HTR6CHRM5MEN1LMNAKMT2A
SCHEMBL4569678 0.84 PTGDR (0.43) PTGDRPTGDR2PKMTSHRHTR6
SCHEMBL1156789 0.83 LMNA (0.39) PTGDR2PKMTSHRCHRM5ALDH1A1
SCHEMBL1156756 0.83 PTGER2 (0.38) PTGDR2TSHRPTGER2ALDH1A1KMT2A
SCHEMBL2418769 0.82 HTR6 (0.37) PTGDRPTGDR2PKMTSHRHTR6
Carbamic Acid SCHEMBL4791646 0.82 PTGER2 (0.39) TSHRPTGER2ALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2114917-A2 PYRROLE COMPOUNDS Takeda Pharmaceutical Company Limited (JP) 2009-11-11 EP disclosed
WO-2008108380-A2 PYRROLE COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2008-09-12 WO disclosed