SCHEMBL4572811

SCHEMBL4572811

CS(=O)(=O)NC(=O)CCc1ccc(N)cc1

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PLA2G10 O15496 1/20 0.44
RECQL P46063 1/20 0.43
GRIN1 Q05586 5/20 0.42
GRIN2B Q13224 5/20 0.42
NR4A2 P43354 1/20 0.42
ALDH1A1 P00352 3/20 0.42
GFER P55789 1/20 0.42
MTNR1A P48039 1/20 0.41
MTNR1B P49286 1/20 0.41
HDAC1 Q13547 2/20 0.41
DHFR P00374 1/20 0.41
TSHR P16473 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
LMNA P02545 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23733121 0.83 HDAC2 (0.59) PLA2G10RECQLNR4A2ALDH1A1HDAC1
SCHEMBL21887555 0.83 PDE4B (0.46) ALDH1A1DHFRTSHRSMN1; SMN2TDP1
SCHEMBL6821715 0.79 GFER (0.48) ALDH1A1GFERHDAC1TSHRTDP1
SCHEMBL2635132 0.77 HDAC1 (0.67) GFERHDAC1HDAC6
SCHEMBL23703229 0.75 PRMT1 (0.60) ALDH1A1HDAC1DHFRTSHRSMN1; SMN2
SCHEMBL29852698 0.75 P4HTM (0.46) PLA2G10NR4A2ALDH1A1MTNR1AMTNR1B
SCHEMBL22403771 0.74 HPGD (0.54) ALDH1A1CA1CA2
Sulfuric Acid SCHEMBL4181579 0.73 IDO1 (0.49) RECQLALDH1A1GFERLMNACA2
SCHEMBL1404834 0.72 ALDH1A1 (0.63) RECQLALDH1A1GFERTSHRSMN1; SMN2
SCHEMBL13806431 0.72 POLB (0.51) ALDH1A1HDAC1LMNAHDAC6CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080114007-A1 5-OXO-5,8-DIHYDRO-PYRIDO-PYRIMIDINES AS INHIBITORS OF C-FMS KINASE JANSSEN PHARMACEUTICA N.V. (BE) 2008-05-15 US disclosed
WO-2008055013-A2 5-OXO-5,8 - DIHYDRO - PYRIDO - PYRIMIDINES AS INHIBITORS OF C-FMS KINASE JANSSEN PHARMACEUTICA N.V. (BE) 2008-05-08 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080114007-A1 5-OXO-5,8-DIHYDRO-PYRIDO-PYRIMIDINES AS INHIBITORS OF C-FMS KINASE FLT3, FES, ALK PLA2G10 3780/4885RECQL 1445/4885GRIN1 3463/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.