SCHEMBL4573136

SCHEMBL4573136

CC(C)(C#N)c1ccc(N2CCNCC2)nc1

nearest known ligand 0.51

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PANK3 Q9H999 2/20 0.44
PLD1 Q13393 1/20 0.43
NTRK1 P04629 1/20 0.41
ADRB1 P08588 1/20 0.40
RET P07949 5/20 0.40
GPR119 Q8TDV5 1/20 0.39
BPTF Q12830 2/20 0.39
KCNH2 Q12809 1/20 0.39
CACNA1C Q13936 1/20 0.39
ASIC3 Q9UHC3 1/20 0.39
HRH4 Q9H3N8 2/20 0.39
ALDH1A1 P00352 1/20 0.38
MAPT P10636 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL28880753 0.99 PANK3 (0.43) PANK3PLD1NTRK1ADRB1RET
Hydrochloric Acid SCHEMBL29978981 0.99 PANK3 (0.43) PANK3PLD1NTRK1ADRB1RET
SCHEMBL270536 0.83 PLD1 (0.49) PANK3PLD1NTRK1ADRB1GPR119
SCHEMBL15316690 0.81 ADRB1 (0.50) PLD1ADRB1GPR119BPTFALDH1A1
SCHEMBL17128345 0.81 OGA (0.50) PANK3PLD1NTRK1ADRB1GPR119
Hydrochloric Acid SCHEMBL28341448 0.79 OGA (0.49) PANK3PLD1NTRK1ADRB1GPR119
SCHEMBL27772210 0.78 ADRB1 (0.48) PLD1ADRB1GPR119ALDH1A1MAPT
SCHEMBL17035908 0.77 ADRB1 (0.60) PLD1ADRB1ALDH1A1MAPT
SCHEMBL30101389 0.77 ADRB1 (0.60) PLD1ADRB1ALDH1A1MAPT
SCHEMBL231823 0.77 ADRB1 (0.60) PLD1ADRB1ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019062657-A1 NITROGEN HETEROCYCLIC DERIVATIVE, PREPARATION METHOD THEREFOR, AND PHARMACEUTICAL USE THEREOF 北京越之康泰生物医药科技有限公司 2019-04-04 WO disclosed
WO-2009001127-A1 CYANOCYCLOPROPYLCARBOXAMIDES AS CATHEPSIN INHIBITORS ASTRAZENECA AB (SE) 2008-12-31 WO disclosed
WO-2009001127-A1 CYANOCYCLOPROPYLCARBOXAMIDES AS CATHEPSIN INHIBITORS ASTRAZENECA AB (SE) 2008-12-31 WO disclosed