SCHEMBL4573351

SCHEMBL4573351

CS(=O)(=O)c1ccc2nc(N3CCNCC3)sc2c1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCN4A P35499 2/20 0.55
SCN9A Q15858 2/20 0.55
NPC1 O15118 9/20 0.53
RAB9A P51151 9/20 0.53
TSHR P16473 1/20 0.48
NPSR1 Q6W5P4 1/20 0.48
POLB P06746 1/20 0.47
CTSL P07711 1/20 0.47
CTSB P07858 1/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2D6 P10635 1/20 0.47
CYP2C9 P11712 1/20 0.47
CTSK P43235 1/20 0.47
APOBEC3A P31941 1/20 0.47
APOBEC3G Q9HC16 1/20 0.47
HTR6 P50406 2/20 0.46
ALDH1A1 P00352 4/20 0.46
SMN1; SMN2 Q16637 3/20 0.46
MAPT P10636 1/20 0.46
HTT P42858 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3232592 0.80 SCN4A (0.61) SCN4ASCN9ANPC1RAB9ANPSR1
SCHEMBL3913015 0.79 HTR6 (0.63) SCN4ASCN9AHTR6
Hydrochloric Acid SCHEMBL4083731 0.78 HTR6 (0.62) SCN4ASCN9AHTR6
SCHEMBL2711602 0.77 RAB9A (0.79) SCN4ASCN9ANPC1RAB9ATSHR
SCHEMBL2710695 0.77 NPC1 (0.76) SCN4ASCN9ANPC1RAB9AALDH1A1
SCHEMBL1981263 0.77 RAB9A (0.76) SCN4ASCN9ANPC1RAB9AAPOBEC3A
SCHEMBL31349392 0.77 NPC1 (0.70) SCN4ASCN9ANPC1RAB9ACYP3A4
SCHEMBL13279558 0.77 AR (0.70) SCN4ASCN9ANPC1RAB9ACYP3A4
SCHEMBL2709859 0.77 NPC1 (0.74) SCN4ASCN9ANPC1RAB9ANPSR1
SCHEMBL3093424 0.77 NPC1 (0.70) SCN4ASCN9ANPC1RAB9ACYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009001127-A1 CYANOCYCLOPROPYLCARBOXAMIDES AS CATHEPSIN INHIBITORS ASTRAZENECA AB (SE) 2008-12-31 WO disclosed
WO-2009001127-A1 CYANOCYCLOPROPYLCARBOXAMIDES AS CATHEPSIN INHIBITORS ASTRAZENECA AB (SE) 2008-12-31 WO disclosed