SCHEMBL4574004

SCHEMBL4574004

CC(=O)NCCCCN1CCN(c2cccc3sccc23)CC1

nearest known ligand 0.61

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 17/20 0.61
HTR2A P28223 17/20 0.61
HTR1A P08908 16/20 0.61
FAAH O00519 1/20 0.60
DRD3 P35462 1/20 0.60
HTR2C P28335 2/20 0.57
ADRA1A P35348 2/20 0.57
HRH1 P35367 2/20 0.57
KCNH2 Q12809 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4574186 0.99 DRD2 (0.60) DRD2HTR2AHTR1AFAAHDRD3
SCHEMBL4624803 0.89 DRD2 (0.58) DRD2HTR2AHTR1AFAAHDRD3
SCHEMBL4575061 0.85 DRD2 (0.61) DRD2HTR2AHTR1AFAAHDRD3
SCHEMBL29433199 0.85 DRD2 (0.75) DRD2HTR2AHTR1AHTR2CADRA1A
SCHEMBL4589842 0.84 HTR1A (0.51) DRD2HTR2AHTR1AFAAHDRD3
SCHEMBL4574007 0.83 DRD2 (0.61) DRD2HTR2AHTR1AHTR2CADRA1A
SCHEMBL294229 0.83 DRD2 (0.66) DRD2HTR2AHTR1ADRD3HTR2C
SCHEMBL30176777 0.81 DRD2 (0.67) DRD2HTR2AHTR1AHTR2CADRA1A
SCHEMBL293734 0.81 DRD2 (0.67) DRD2HTR2AHTR1AHTR2CADRA1A
SCHEMBL4574005 0.81 DRD2 (0.64) DRD2HTR2AHTR1AHTR2CADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008047883-A1 PIPERAZINE-SUBSTITUTED BENZOTHIOPHENES FOR TREATMENT OF MENTAL DISORDERS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2008-04-24 WO claimed
WO-2008047883-A1 PIPERAZINE-SUBSTITUTED BENZOTHIOPHENES FOR TREATMENT OF MENTAL DISORDERS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2008-04-24 WO disclosed