SCHEMBL4574387

SCHEMBL4574387

C[C@@H]1CN(Cc2cccc(F)c2F)CCN1

nearest known ligand 0.44

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 2/20 0.44
JAK3 P52333 2/20 0.44
MLNR O43193 13/20 0.41
GAA P10253 1/20 0.41
JAK1 P23458 1/20 0.41
TYK2 P29597 1/20 0.41
CYP3A4 P08684 2/20 0.40
CYP2D6 P10635 1/20 0.40
KCNH2 Q12809 1/20 0.40
ALDH1A1 P00352 1/20 0.40
CHRM2 P08172 2/20 0.39
CHRM1 P11229 2/20 0.39
CHRM3 P20309 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2022959 0.80 XIAP (0.40) MLNRCYP3A4
SCHEMBL2925434 0.79 LMNA (0.54) GAAALDH1A1CHRM2
SCHEMBL14708215 0.78 JAK2 (0.52) JAK2JAK3GAAJAK1TYK2
SCHEMBL25640506 0.78 TACR1 (0.39) JAK2JAK3GAAJAK1TYK2
SCHEMBL20817868 0.78 LMNA (0.62) MLNRALDH1A1
SCHEMBL30616176 0.78 LMNA (0.62) MLNRALDH1A1
SCHEMBL13595851 0.77 ACHE (0.61) CYP2D6
SCHEMBL4590018 0.77 XIAP (0.48) MLNRCYP3A4
SCHEMBL4590022 0.77 XIAP (0.48) MLNRCYP3A4
SCHEMBL3172097 0.77 KDM4E (0.55) MLNRALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008134035-A1 ALPHA-UNSUBSTITUTED ARYLMETHYL PIPERAZINE PYRAZOLO[1,5-A] PYRIMIDINE AMIDE DERIVATIVES PANACOS PHARMACEUTICALS, INC. (US) 2008-11-06 WO disclosed