SCHEMBL4574455

SCHEMBL4574455

Fc1cc(F)c(F)c(CN2CCNCC2)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
LMNA P02545 1/20 0.42
SLC6A4 P31645 3/20 0.42
CHRM2 P08172 2/20 0.42
CYP1A2 P05177 1/20 0.42
OPRD1 P41143 1/20 0.42
OPRK1 P41145 1/20 0.42
SLC6A2 P23975 2/20 0.41
KCNH2 Q12809 2/20 0.41
SLC6A3 Q01959 1/20 0.41
APOBEC3A P31941 1/20 0.41
CTDSP1 Q9GZU7 1/20 0.41
APOBEC3G Q9HC16 1/20 0.41
SIGMAR1 Q99720 1/20 0.41
SOS1 Q07889 3/20 0.38
CXCR4 P61073 2/20 0.38
MEN1 O00255 1/20 0.38
CHRM1 P11229 1/20 0.38
ADRA2C P18825 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2922854 0.79 KDM4E (0.51) KDM4ESMN1; SMN2LMNASLC6A4CHRM2
SCHEMBL2924537 0.79 KDM4E (0.70) KDM4ESMN1; SMN2LMNASLC6A4CHRM2
SCHEMBL2022959 0.79 XIAP (0.40)
SCHEMBL14013388 0.78 SCN9A (0.36) KDM4ESMN1; SMN2LMNAKCNH2
SCHEMBL4573863 0.78 SCN9A (0.36) KDM4ESMN1; SMN2LMNAKCNH2
Hydrochloric Acid SCHEMBL1238937 0.78 KDM4E (0.68) KDM4ESMN1; SMN2LMNASLC6A4CHRM2
Hydrochloric Acid SCHEMBL15568255 0.78 KDM4E (0.68) KDM4ESMN1; SMN2LMNASLC6A4CHRM2
SCHEMBL4574934 0.77 KDM4E (0.34) KDM4ESMN1; SMN2
SCHEMBL4574383 0.77 RIPK1 (0.34) KDM4ESMN1; SMN2
SCHEMBL14303254 0.77 LMNA (0.46) KDM4ESMN1; SMN2LMNASLC6A4CHRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008134035-A1 ALPHA-UNSUBSTITUTED ARYLMETHYL PIPERAZINE PYRAZOLO[1,5-A] PYRIMIDINE AMIDE DERIVATIVES PANACOS PHARMACEUTICALS, INC. (US) 2008-11-06 WO disclosed
WO-2008134035-A1 ALPHA-UNSUBSTITUTED ARYLMETHYL PIPERAZINE PYRAZOLO[1,5-A] PYRIMIDINE AMIDE DERIVATIVES PANACOS PHARMACEUTICALS, INC. (US) 2008-11-06 WO disclosed