SCHEMBL4574508

SCHEMBL4574508

C=CCOc1cc(C(=O)OCC)cn2c(C)c(C)nc12

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.39
SMN1; SMN2 Q16637 3/20 0.39
ALDH1A1 P00352 3/20 0.38
HSD17B2 P37059 1/20 0.37
MAPK1 P28482 3/20 0.37
RAB9A P51151 2/20 0.37
HCRTR1 O43613 1/20 0.37
TP53 P04637 1/20 0.37
MAPT P10636 1/20 0.37
ALOX15 P16050 1/20 0.37
PSEN1 P49768 1/20 0.37
PSEN2 P49810 1/20 0.37
APH1B Q8WW43 1/20 0.37
NCSTN Q92542 1/20 0.37
APH1A Q96BI3 1/20 0.37
PSENEN Q9NZ42 1/20 0.37
HPGD P15428 2/20 0.36
HSD17B10 Q99714 2/20 0.36
CYP3A4 P08684 2/20 0.36
CYP2C9 P11712 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5566371 0.84 KDM4E (0.36) KDM4ESMN1; SMN2ALDH1A1MAPTHSD17B10
SCHEMBL4591398 0.80 ATP4A (0.47) SMN1; SMN2ALDH1A1MAPK1RAB9AHCRTR1
SCHEMBL4573822 0.78 CA12 (0.48) KDM4ESMN1; SMN2ALDH1A1HSD17B2MAPK1
SCHEMBL4169299 0.77 SMN1; SMN2 (0.44) KDM4ESMN1; SMN2ALDH1A1MAPK1RAB9A
Alcohol SCHEMBL5566652 0.76 CA12 (0.46) KDM4ESMN1; SMN2ALDH1A1HSD17B2MAPK1
SCHEMBL8546144 0.73 KDM4E (0.48) KDM4ESMN1; SMN2ALDH1A1HSD17B2HPGD
SCHEMBL12126791 0.71 HSD17B2 (0.55) KDM4ESMN1; SMN2ALDH1A1HSD17B2RAB9A
SCHEMBL6580057 0.71 HSD17B2 (0.67) KDM4EALDH1A1HSD17B2TP53MAPT
SCHEMBL5152746 0.71 HSD17B2 (0.51) KDM4EHSD17B2
SCHEMBL4737793 0.70 KDM4E (0.41) KDM4EALDH1A1HSD17B2RAB9AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008071766-A2 SPIRO-INDENE SUBSTITUTED IMIDAZONAPHYTHYRIDINE AND PYRANOIMIDAZOPYRIDINE DERIVATIVES AS INHIBITORS OF GASTRIC ACID SECRETION NYCOMED GMBH (DE) 2008-06-19 WO disclosed