SCHEMBL4575162

SCHEMBL4575162

COc1ccc(Nc2ccc(Cl)cc2)c([N+](=O)[O-])c1

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 4/20 0.70
AKR1C2 P52895 4/20 0.70
MAPT P10636 8/20 0.69
L3MBTL1 Q9Y468 3/20 0.69
MAPK1 P28482 3/20 0.69
TDP1 Q9NUW8 3/20 0.69
ALDH1A1 P00352 1/20 0.69
ALDH3A1 P30838 1/20 0.62
AKR1B10 O60218 1/20 0.59
AKR1B1 P15121 1/20 0.59
AKR1C4 P17516 1/20 0.59
AKR1C1 Q04828 1/20 0.59
LMNA P02545 4/20 0.58
MEN1 O00255 3/20 0.58
KMT2A Q03164 3/20 0.58
POLB P06746 2/20 0.58
GAA P10253 2/20 0.56
HTT P42858 1/20 0.56
SMN1; SMN2 Q16637 3/20 0.55
CYP3A4 P08684 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4932340 0.92 MAPT (0.73) AKR1C3AKR1C2MAPTL3MBTL1MAPK1
SCHEMBL2328384 0.89 MAPT (0.58) AKR1C3AKR1C2MAPTL3MBTL1MAPK1
SCHEMBL14656691 0.87 MAPT (0.84) AKR1C3AKR1C2MAPTL3MBTL1MAPK1
SCHEMBL11516026 0.86 AKR1C3 (0.70) AKR1C3AKR1C2MAPTL3MBTL1MAPK1
SCHEMBL6179431 0.86 AKR1C3 (0.74) AKR1C3AKR1C2MAPTL3MBTL1MAPK1
SCHEMBL11383159 0.84 L3MBTL1 (0.82) MAPTL3MBTL1MAPK1TDP1ALDH1A1
SCHEMBL4744863 0.83 MAPT (0.64) AKR1C3AKR1C2MAPTL3MBTL1MAPK1
SCHEMBL9121900 0.83 MAPT (0.65) AKR1C3AKR1C2MAPTL3MBTL1MAPK1
SCHEMBL4933766 0.82 MAPT (0.67) AKR1C3AKR1C2MAPTL3MBTL1MAPK1
SCHEMBL2309318 0.82 MAPT (1.00) AKR1C3AKR1C2MAPTL3MBTL1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008107322-A1 INDOLE, BENZIMIDAZOLE OR BENZOTRIAZOLE DERIVATIVES INCLUDING A PIPERIDINE OR PIPERAZINE CORE AS ANTI-NEOPLASIC AGENTS OR CELL PROLIFERATION INHIBITORS CEREP (FR) 2008-09-12 WO disclosed