SCHEMBL45780

SCHEMBL45780

CN(C)C(=O)c1ccc2c(c1)CCCN2

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.68
MAPT P10636 2/20 0.68
ALDH1A1 P00352 4/20 0.48
GAA P10253 2/20 0.48
ALOX15 P16050 2/20 0.48
LMNA P02545 1/20 0.48
TP53 P04637 1/20 0.48
THRB P10828 1/20 0.48
CASP1 P29466 1/20 0.48
HTT P42858 1/20 0.48
CASP7 P55210 1/20 0.48
HSD17B10 Q99714 1/20 0.48
TDP1 Q9NUW8 1/20 0.48
CA12 O43570 1/20 0.47
CA1 P00915 1/20 0.47
CA2 P00918 1/20 0.47
CA9 Q16790 1/20 0.47
PLAU P00749 1/20 0.44
PIR O00625 1/20 0.43
GSK3B P49841 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8511891 0.91 KDM4E (0.54) KDM4EMAPTALDH1A1ALOX15ACHE
SCHEMBL6983698 0.84 KDM4E (0.62) KDM4EMAPTALDH1A1GAAALOX15
SCHEMBL6986243 0.84 KDM4E (0.62) KDM4EMAPTALDH1A1GAAALOX15
SCHEMBL3096482 0.83 MAPT (0.73) KDM4EMAPTALDH1A1GAAALOX15
SCHEMBL29673258 0.81 KDM4E (1.00) KDM4EMAPTALDH1A1GAAALOX15
SCHEMBL45202 0.81 KDM4E (1.00) KDM4EMAPTALDH1A1GAAALOX15
SCHEMBL28039955 0.80 MAPT (0.73) KDM4EMAPTALDH1A1GAAALOX15
SCHEMBL12486871 0.80 KDM4E (0.73) KDM4EMAPTALDH1A1GAAALOX15
SCHEMBL30011603 0.80 KDM4E (0.73) KDM4EMAPTALDH1A1GAAALOX15
SCHEMBL29995197 0.79 MAPT (0.68) KDM4EMAPTALDH1A1GAAALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2588458-A1 NOVEL TETRAHYDROQUINOLINE DERIVATIVES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-08 EP claimed
WO-2012001020-A1 NOVEL TETRAHYDROQUINOLINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-05 WO claimed
EP-4381284-B1 LIGAND-TARGET INTERACTION ANALYSIS BY PHOTOCHEMICALLY INDUCED DYNAMIC NUCLEAR POLARIZATION (PHOTO-CIDNP) ENHANCED NMR SPECTROSCOPY ETH ZUERICH (CH) 2025-07-09 EP disclosed
US-20240345008-A1 LIGAND-TARGET INTERACTION ANALYSIS BY PHOTOCHEMICALLY INDUCED DYNAMIC NUCLEAR POLARIZATION (PHOTO-CIDNP) ENHANCED NMR SPECTROSCOPY ETH ZURICH (CH) 2024-10-17 US disclosed
EP-2588458-A1 NOVEL TETRAHYDROQUINOLINE DERIVATIVES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-08 EP disclosed
WO-2012001020-A1 NOVEL TETRAHYDROQUINOLINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-05 WO disclosed