SCHEMBL4580481

SCHEMBL4580481

Cc1ccc(S(=O)(=O)NCCN(C(C)C(NS(=O)(=O)c2ccc(C)cc2)c2ccc([N+](=O)[O-])cc2)S(=O)(=O)c2ccc(C)cc2)cc1

nearest known ligand 0.51

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 5/20 0.51
KMT2A Q03164 5/20 0.51
RAB9A P51151 1/20 0.51
ALDH1A1 P00352 7/20 0.49
MAPT P10636 3/20 0.49
GAA P10253 1/20 0.49
CA9 Q16790 2/20 0.43
HTT P42858 2/20 0.42
PKM P14618 1/20 0.42
TSHR P16473 1/20 0.41
CA2 P00918 2/20 0.40
CA12 O43570 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2C19 P33261 1/20 0.40
ALOX15 P16050 1/20 0.40
CA1 P00915 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4094207 0.77 MEN1 (0.53) MEN1KMT2ARAB9AALDH1A1MAPT
SCHEMBL9906204 0.73 MEN1 (0.52) MEN1KMT2ARAB9AALDH1A1MAPT
SCHEMBL10683290 0.73 ALDH1A1 (0.65) MEN1KMT2ARAB9AALDH1A1MAPT
SCHEMBL29168805 0.72 ALDH1A1 (0.48) MEN1KMT2ARAB9AALDH1A1MAPT
SCHEMBL598734 0.71 MEN1 (0.55) MEN1KMT2ARAB9AALDH1A1MAPT
SCHEMBL7035347 0.70 TSHR (0.65) MEN1KMT2ARAB9AALDH1A1MAPT
SCHEMBL6801249 0.69 ALDH1A1 (0.77) MEN1KMT2ARAB9AALDH1A1MAPT
SCHEMBL17793710 0.69 KMT2A (0.61) MEN1KMT2ARAB9AALDH1A1MAPT
SCHEMBL12478115 0.69 KMT2A (0.57) MEN1KMT2ARAB9AALDH1A1MAPT
SCHEMBL10737899 0.68 TRPV4 (0.49) CA9CA2CA12CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2004642-A1 BIFUNCTIONAL POLYAZAMACROCYCLIC CHELATING AGENTS MDS (Canada) Inc. (CA) 2008-12-24 EP disclosed
WO-2007104135-A1 BIFUNCTIONAL POLYAZAMACROCYCLIC CHELATING AGENTS MDS (CANADA) INC. (CA) 2007-09-20 WO disclosed