SCHEMBL4582141

SCHEMBL4582141

Cc1n[nH]c(=O)c(-c2c(F)cccc2F)c1-c1nccs1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 2/20 0.42
ADORA1 P30542 2/20 0.42
MGAM O43451 1/20 0.34
GAA P10253 1/20 0.34
SI P14410 1/20 0.34
MGAM2 Q2M2H8 1/20 0.34
CHEK1 O14757 1/20 0.34
NTRK1 P04629 1/20 0.34
MAT2A P31153 1/20 0.33
PDPK1 O15530 1/20 0.33
HCRTR1 O43613 1/20 0.33
HCRTR2 O43614 1/20 0.33
ALK Q9UM73 3/20 0.33
INSR P06213 2/20 0.33
TYK2 P29597 1/20 0.33
ILK Q13418 1/20 0.33
PARP1 P09874 2/20 0.32
PARP2 Q9UGN5 2/20 0.32
PARP3 Q9Y6F1 1/20 0.32
KMT2A Q03164 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4582860 0.76 NPC1 (0.39) CHEK1DRD1
SCHEMBL10015937 0.75 AKT2 (0.51) CHEK1TYK2KMT2A
SCHEMBL28020115 0.75 PDPK1 (0.50) ADORA2AADORA1MGAMGAASI
SCHEMBL2351250 0.72 NPC1 (0.40) GAACHEK1TYK2PARP2KMT2A
SCHEMBL4582362 0.71 ADORA2A (0.41) ADORA2APARP1KMT2A
SCHEMBL3617725 0.69 TYMP (0.39) GAACHEK1ILKKMT2A
SCHEMBL2248431 0.68 PDPK1 (0.43) ADORA2AADORA1MGAMGAASI
SCHEMBL11402984 0.68 PTGES (0.44) ADORA2AADORA1MGAMGAASI
SCHEMBL16254413 0.68 SRD5A1 (0.31) PARP1
SCHEMBL10446010 0.68 PDPK1 (0.40) MGAMGAASIMGAM2PDPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1972623-A1 Arylpyridazines as fungicides Bayer CropScience AG (DE) 2008-09-24 EP disclosed