SCHEMBL4584319

SCHEMBL4584319

COC1CN(C(=O)c2cc3c(s2)CN(C)CC3)CC1NC(=O)Oc1ccc(Cl)s1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
F10 P00742 9/20 0.44
WDR91 A4D1P6 1/20 0.39
ALDH1A1 P00352 3/20 0.35
HPGD P15428 2/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2C19 P33261 1/20 0.35
HDAC6 Q9UBN7 2/20 0.35
MCHR1 Q99705 1/20 0.33
L3MBTL1 Q9Y468 2/20 0.33
PARP1 P09874 1/20 0.33
PARP2 Q9UGN5 1/20 0.33
ESR1 P03372 1/20 0.33
POLB P06746 1/20 0.33
MAPT P10636 1/20 0.33
NR4A1 P22736 1/20 0.33
KMT2A Q03164 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
PRMT5 O14744 1/20 0.32
WDR77 Q9BQA1 1/20 0.32
DNMT1 P26358 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4583142 0.93 F10 (0.44) F10WDR91ALDH1A1HPGDCYP1A2
SCHEMBL8509610 0.88 F10 (0.47) F10WDR91HDAC6KMT2A
SCHEMBL3306401 0.88 F10 (0.47) F10WDR91HDAC6KMT2A
SCHEMBL13372904 0.88 F10 (0.44) F10WDR91ALDH1A1HPGDCYP1A2
SCHEMBL4435127 0.88 F10 (0.32) F10ALDH1A1HPGDCYP1A2CYP2C19
SCHEMBL4436378 0.86 ALDH1A1 (0.33) F10ALDH1A1HPGDCYP1A2CYP2C19
SCHEMBL4583647 0.85 F10 (0.38) F10HDAC6MCHR1POLBMAPT
SCHEMBL4433466 0.85 F10 (0.32) F10
SCHEMBL4432476 0.85 F10 (0.42) F10HDAC6MCHR1MAPTPRMT5
SCHEMBL13372905 0.84 F10 (0.33) F10ALDH1A1HPGDCYP1A2CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2132193-B1 SUBSTITUTED PYRROLIDINE AMIDES, THE PRODUCTION THEREOF, AND THE USE THEREOF AS MEDICATIONS BOEHRINGER INGELHEIM INT (DE) 2012-10-24 EP disclosed
EP-1975165-A1 Substituted pyrrolidinamides, their production and utilisation as medicine Boehringer Ingelheim Pharma GmbH & Co. KG (DE) 2008-10-01 EP disclosed