SCHEMBL4585686

SCHEMBL4585686

CNc1c(C(=O)O)cnc2ccc(C=C3SC(Nc4cc(NC(=O)C5CCC5)ccc4Cl)=NC3=O)cc12

nearest known ligand 0.39

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
EGFR P00533 10/20 0.39
MELK Q14680 4/20 0.34
CISD1 Q9NZ45 1/20 0.33
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
GAA P10253 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4585672 1.00 EGFR (0.39) EGFRMELKCISD1KDM4EALDH1A1
SCHEMBL5050823 0.91 MAPT (0.41) EGFRKDM4EALDH1A1GAASMN1; SMN2
SCHEMBL2989487 0.91 MAPT (0.41) EGFRKDM4EALDH1A1GAASMN1; SMN2
SCHEMBL2989491 0.86 EGFR (0.34) EGFRCISD1KDM4EALDH1A1GAA
SCHEMBL2988900 0.83 EGFR (0.40) EGFRCISD1L3MBTL1
SCHEMBL2988902 0.83 EGFR (0.40) EGFRCISD1L3MBTL1
Trifluoroacetic Acid SCHEMBL4586199 0.83 GBA1 (0.39) EGFRMELKKDM4EALDH1A1
Trifluoroacetic Acid SCHEMBL4586182 0.83 GBA1 (0.39) EGFRMELKKDM4EALDH1A1
SCHEMBL4586161 0.82 PTGDR2 (0.34) EGFRCISD1L3MBTL1
SCHEMBL4586168 0.82 PTGDR2 (0.34) EGFRCISD1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1879563-A4 NOVEL CHEMICAL COMPOUNDS SMITHKLINE BEECHAM CORP (US) 2008-07-16 EP disclosed
EP-1879563-A2 NOVEL CHEMICAL COMPOUNDS Smithkline Beecham Corporation (US) 2008-01-23 EP disclosed
WO-2006132739-A2 NOVEL CHEMICAL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2006-12-14 WO disclosed