SCHEMBL4586161

SCHEMBL4586161

CCc1nc2ccc(/C=C3\SC(Nc4cc(NC(=O)C5CCC5)ccc4Cl)=NC3=O)cc2cc1C(=O)O

nearest known ligand 0.35

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 3/20 0.34
EGFR P00533 3/20 0.34
GBA1 P04062 1/20 0.34
NR2E3 Q9Y5X4 2/20 0.33
CISD1 Q9NZ45 1/20 0.33
ABL1 P00519 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
MCHR1 Q99705 2/20 0.32
HDAC4 P56524 1/20 0.32
ENPP2 Q13822 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4586168 1.00 PTGDR2 (0.34) PTGDR2EGFRGBA1NR2E3CISD1
Trifluoroacetic Acid SCHEMBL2991042 0.96 EGFR (0.33) PTGDR2EGFRGBA1NR2E3CISD1
Trifluoroacetic Acid SCHEMBL2991046 0.96 EGFR (0.33) PTGDR2EGFRGBA1NR2E3CISD1
SCHEMBL4587397 0.87 ALDH1A1 (0.38) PTGDR2NR2E3CISD1MCHR1HDAC4
SCHEMBL4587403 0.87 ALDH1A1 (0.38) PTGDR2NR2E3CISD1MCHR1HDAC4
SCHEMBL2989491 0.87 EGFR (0.34) PTGDR2EGFRGBA1NR2E3CISD1
Trifluoroacetic Acid SCHEMBL2995750 0.83 ALDH1A1 (0.35) CISD1
Trifluoroacetic Acid SCHEMBL2995754 0.83 ALDH1A1 (0.35) CISD1
Trifluoroacetic Acid SCHEMBL2994088 0.83 GBA1 (0.34) PTGDR2EGFRGBA1CISD1MCHR1
SCHEMBL4585672 0.82 EGFR (0.39) EGFRCISD1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1879563-A4 NOVEL CHEMICAL COMPOUNDS SMITHKLINE BEECHAM CORP (US) 2008-07-16 EP claimed
EP-1879563-A2 NOVEL CHEMICAL COMPOUNDS Smithkline Beecham Corporation (US) 2008-01-23 EP claimed
WO-2006132739-A2 NOVEL CHEMICAL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2006-12-14 WO claimed