SCHEMBL2989491

SCHEMBL2989491

CCc1nc2ccc(C=C3SC(Nc4cc(NC(=O)C5CCC5)ccc4Cl)=NC3=O)cc2c(NC)c1C(=O)O

nearest known ligand 0.34

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
EGFR P00533 5/20 0.34
GBA1 P04062 2/20 0.34
PTGDR2 Q9Y5Y4 3/20 0.33
CISD1 Q9NZ45 1/20 0.32
GLA P06280 1/20 0.32
MCHR1 Q99705 2/20 0.32
ABL1 P00519 1/20 0.31
KDM4E B2RXH2 2/20 0.31
ALDH1A1 P00352 1/20 0.31
GAA P10253 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
MEN1 O00255 1/20 0.31
POLB P06746 1/20 0.31
KMT2A Q03164 1/20 0.31
NR2E3 Q9Y5X4 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL2994088 0.87 GBA1 (0.34) EGFRGBA1PTGDR2CISD1GLA
SCHEMBL4586168 0.87 PTGDR2 (0.34) EGFRGBA1PTGDR2CISD1MCHR1
SCHEMBL4586161 0.87 PTGDR2 (0.34) EGFRGBA1PTGDR2CISD1MCHR1
SCHEMBL4585672 0.86 EGFR (0.39) EGFRCISD1KDM4EALDH1A1GAA
SCHEMBL4585686 0.86 EGFR (0.39) EGFRCISD1KDM4EALDH1A1GAA
Trifluoroacetic Acid SCHEMBL2995877 0.86 FABP3 (0.35) EGFRGBA1CISD1MCHR1
Trifluoroacetic Acid SCHEMBL2988931 0.84 GBA1 (0.39) EGFRGBA1GLAMCHR1KDM4E
SCHEMBL2989487 0.84 MAPT (0.41) EGFRKDM4EALDH1A1GAASMN1; SMN2
SCHEMBL5050823 0.84 MAPT (0.41) EGFRKDM4EALDH1A1GAASMN1; SMN2
Trifluoroacetic Acid SCHEMBL2991042 0.83 EGFR (0.33) EGFRGBA1PTGDR2CISD1MCHR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080214455-A1 Novel Chemical Compounds SMITHKLINE BEECHAM CORPORATION 2008-09-04 US claimed
US-20100184774-A1 METHODS OF TREATMENT SMITHKLINE BEECHAM CORPORATION 2010-07-22 US disclosed
EP-2164494-A1 METHODS OF TREATMENT GlaxoSmithKline LLC (US) 2010-03-24 EP disclosed
WO-2008150837-A1 METHODS OF TREATMENT SMITHKLINE BEECHAM CORPORATION (US) 2008-12-11 WO disclosed
US-20080214455-A1 Novel Chemical Compounds SMITHKLINE BEECHAM CORPORATION 2008-09-04 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080214455-A1 Novel Chemical Compounds HIPK3, HIPK1, HIPK4 EGFR 4159/4885GBA1 487/4885PTGDR2 4536/4885
US-20100184774-A1 METHODS OF TREATMENT OPRL1, BRCA1, PKD1 EGFR 2273/4885GBA1 606/4885PTGDR2 408/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.