SCHEMBL4585928

SCHEMBL4585928

Clc1ccsc1-c1nc(N2CCNCC2)no1

nearest known ligand 0.50

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CASP3 P42574 15/20 0.50
HTR2C P28335 2/20 0.47
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44
SCN9A Q15858 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4585637 0.88 NPC1 (0.57) CASP3NPC1RAB9A
SCHEMBL4424692 0.86 RAB9A (0.59) CASP3NPC1RAB9A
SCHEMBL4593631 0.85 CASP3 (0.51) CASP3NPC1RAB9A
SCHEMBL4593399 0.82 CASP3 (0.48) CASP3NPC1RAB9A
SCHEMBL4593834 0.80 CASP3 (0.49) CASP3NPC1RAB9A
SCHEMBL4588636 0.76 CASP3 (0.44) CASP3NPC1RAB9A
SCHEMBL2248381 0.76 NPC1 (0.75) NPC1RAB9A
SCHEMBL389135 0.74 GBA1 (0.43) CASP3
Trifluoroacetic Acid SCHEMBL4586889 0.73 CASP3 (0.43) CASP3NPC1RAB9A
SCHEMBL4593010 0.72 CASP3 (0.45) CASP3NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1581213-A4 3,5-DISUBSTITUTED- 1,2,4 -OXADIAZOLES AND ANALOGS AS AC TIVATORS OF CASPASES AND INDUCERS OF APOPTOSIS AND THE USE THEREOF CYTOVIA INC (US) 2008-11-19 EP claimed
EP-1581213-A1 3,5-DISUBSTITUTED- 1,2,4 -OXADIAZOLES AND ANALOGS AS AC TIVATORS OF CASPASES AND INDUCERS OF APOPTOSIS AND THE USE THEREOF Cytovia, Inc. (US) 2005-10-05 EP claimed
WO-2004058253-A1 3,5-DISUBSTITUTED-[1,2,4]-OXADIAZOLES AND ANALOGS AS ACTIVATORS OF CASPASES AND INDUCERS OF APOPTOSIS AND THE USE THEREOF CYTOVIA, INC. (US) 2004-07-15 WO claimed