SCHEMBL4586039

SCHEMBL4586039

COC(=O)/C=C/c1ccc(N(Cc2cc(C#N)ccc2F)C2CCN(CCC(C)N)CC2)cc1

nearest known ligand 0.40

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PGR P06401 5/20 0.40
CYP2D6 P10635 4/20 0.40
CYP2C9 P11712 4/20 0.40
DRD2 P14416 3/20 0.39
DRD3 P35462 3/20 0.39
CCR5 P51681 5/20 0.37
NR1H4 Q96RI1 4/20 0.37
HTR2A P28223 1/20 0.36
HTR1D P28221 1/20 0.36
MCHR1 Q99705 1/20 0.35
CFD P00746 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4243356 0.87 CCR5 (0.45) PGRCYP2D6CYP2C9CCR5NR1H4
SCHEMBL4243359 0.87 CCR5 (0.45) PGRCYP2D6CYP2C9CCR5NR1H4
SCHEMBL4586706 0.85 CCR5 (0.40) PGRCYP2D6CYP2C9DRD2DRD3
SCHEMBL4586037 0.84 PGR (0.42) PGRCYP2D6CYP2C9CCR5MCHR1
SCHEMBL4241306 0.82 PGR (0.45) PGRCYP2D6CYP2C9NR1H4
SCHEMBL4241304 0.82 PGR (0.45) PGRCYP2D6CYP2C9NR1H4
SCHEMBL4241217 0.78 CCR5 (0.56) CCR5
SCHEMBL4241224 0.78 CCR5 (0.56) CCR5
SCHEMBL4585509 0.78 CCR5 (0.38) PGRCYP2D6CYP2C9DRD2DRD3
SCHEMBL4586507 0.75 CCR5 (0.43) PGRCYP2D6CYP2C9CCR5HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1708703-A4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC (CA) 2008-04-09 EP disclosed
EP-1708703-A2 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2006-10-11 EP disclosed
WO-2005059107-A2 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2005-06-30 WO disclosed