SCHEMBL4586474

SCHEMBL4586474

O=C1N=C(Nc2c(Cl)cccc2Cl)S/C1=C/c1ccc2nccc(N3CCCCC3)c2c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 6/20 0.41
ALDH1A1 P00352 2/20 0.41
HTT P42858 2/20 0.41
MAPT P10636 2/20 0.41
CHKA P35790 1/20 0.39
MEN1 O00255 5/20 0.39
RAB9A P51151 2/20 0.38
HTR6 P50406 1/20 0.38
ENPP2 Q13822 1/20 0.38
PKM P14618 1/20 0.38
ALOX15 P16050 1/20 0.38
CASP1 P29466 1/20 0.38
HSD17B10 Q99714 1/20 0.38
CLK1 P49759 2/20 0.37
CLK2 P49760 2/20 0.37
DYRK1A Q13627 2/20 0.37
DYRK3 O43781 1/20 0.37
CSNK1E P49674 1/20 0.37
CLK3 P49761 1/20 0.37
GSK3B P49841 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4586479 1.00 KMT2A (0.41) KMT2AALDH1A1HTTMAPTCHKA
SCHEMBL2995679 0.99 KMT2A (0.41) KMT2AALDH1A1HTTMAPTCHKA
SCHEMBL4585273 0.99 KMT2A (0.41) KMT2AALDH1A1HTTMAPTCHKA
SCHEMBL2995682 0.99 KMT2A (0.41) KMT2AALDH1A1HTTMAPTCHKA
Trifluoroacetic Acid SCHEMBL4586308 0.93 CISD1 (0.36) KMT2AALDH1A1HTTMAPTCHKA
Trifluoroacetic Acid SCHEMBL2995171 0.93 CISD1 (0.36) KMT2AALDH1A1HTTMAPTCHKA
Trifluoroacetic Acid SCHEMBL2995167 0.93 CISD1 (0.36) KMT2AALDH1A1HTTMAPTCHKA
SCHEMBL2993546 0.91 MEN1 (0.40) KMT2AALDH1A1HTTMAPTMEN1
SCHEMBL2993532 0.91 HTR6 (0.47) HTR6CLK1CLK2DYRK1ADYRK3
SCHEMBL2996092 0.91 ENPP2 (0.48) HTR6ENPP2CLK1CLK2DYRK1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1879563-A4 NOVEL CHEMICAL COMPOUNDS SMITHKLINE BEECHAM CORP (US) 2008-07-16 EP disclosed
EP-1879563-A2 NOVEL CHEMICAL COMPOUNDS Smithkline Beecham Corporation (US) 2008-01-23 EP disclosed
WO-2006132739-A2 NOVEL CHEMICAL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2006-12-14 WO disclosed