SCHEMBL458675

SCHEMBL458675

Cc1cc(-c2c(Oc3cccc(F)c3)nn3ccnc3c2S(C)(=O)=O)ccc1C(=O)NC1CC1

nearest known ligand 0.44

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
TTK P33981 12/20 0.44
CYP3A4 P08684 3/20 0.44
KCNH2 Q12809 1/20 0.39
PDE4B Q07343 6/20 0.38
CNR1 P21554 1/20 0.37
CNR2 P34972 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL457865 0.76 TTK (0.52) TTK
SCHEMBL458676 0.75 TTK (0.48) TTKCYP3A4
SCHEMBL470200 0.75 TTK (0.55) TTKCYP3A4
SCHEMBL459012 0.71 TTK (0.46) TTKCNR1CNR2
SCHEMBL17416416 0.70 TTK (0.61) TTKCYP3A4
SCHEMBL10279545 0.70 TTK (0.61) TTKCYP3A4
SCHEMBL17416415 0.70 TTK (0.46) TTK
SCHEMBL463296 0.69 TTK (0.55) TTKCYP3A4
SCHEMBL17416371 0.69 TTK (0.60) TTKCYP3A4
SCHEMBL458141 0.69 TTK (0.61) TTKCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2614063-A1 SUBSTITUTED IMIDAZOPYRIDAZINES Bayer Intellectual Property GmbH (DE) 2013-07-17 EP disclosed
WO-2012032031-A1 SUBSTITUTED IMIDAZOPYRIDAZINES BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2012-03-15 WO disclosed