SCHEMBL458676

SCHEMBL458676

Cc1cc(-c2cn3nc(Oc4cccc(F)c4)cc(S(C)(=O)=O)c3n2)ccc1C(=O)NC1CC1

nearest known ligand 0.48

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
TTK P33981 17/20 0.48
CYP3A4 P08684 4/20 0.48
HPGDS O60760 1/20 0.40
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
NTRK1 P04629 1/20 0.37
KDM4E B2RXH2 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL470200 0.84 TTK (0.55) TTKCYP3A4
SCHEMBL458675 0.75 TTK (0.44) TTKCYP3A4
SCHEMBL457866 0.74 TTK (0.54) TTK
SCHEMBL459013 0.73 TTK (0.48) TTK
SCHEMBL17416416 0.73 TTK (0.61) TTKCYP3A4
SCHEMBL10279545 0.73 TTK (0.61) TTKCYP3A4
SCHEMBL463296 0.72 TTK (0.55) TTKCYP3A4
SCHEMBL17416371 0.72 TTK (0.60) TTKCYP3A4
SCHEMBL458141 0.71 TTK (0.61) TTKCYP3A4
SCHEMBL15555488 0.71 TTK (0.63) TTKCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2614063-A1 SUBSTITUTED IMIDAZOPYRIDAZINES Bayer Intellectual Property GmbH (DE) 2013-07-17 EP disclosed
WO-2012032031-A1 SUBSTITUTED IMIDAZOPYRIDAZINES BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2012-03-15 WO disclosed