SCHEMBL4586762

SCHEMBL4586762

Oc1cc(Cl)ccc1Oc1cc(Cl)cc(Cl)c1

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TTR P02766 5/20 0.63
MAPT P10636 2/20 0.63
HPGD P15428 2/20 0.63
NR1I2 O75469 1/20 0.63
LMNA P02545 1/20 0.63
PGR P06401 1/20 0.63
HSP90AA1 P07900 1/20 0.63
ADORA3 P0DMS8 1/20 0.63
HSPA5 P11021 1/20 0.63
CBR1 P16152 1/20 0.63
TBXA2R P21731 1/20 0.63
SLC6A2 P23975 1/20 0.63
AGTR1 P30556 1/20 0.63
SLC6A3 Q01959 1/20 0.63
ALDH1A1 P00352 2/20 0.45
CYP3A4 P08684 2/20 0.45
TSHR P16473 1/20 0.45
HSD17B10 Q99714 1/20 0.45
TDP1 Q9NUW8 1/20 0.45
CYP1A2 P05177 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Soneclosan SCHEMBL29359126 0.86 TTR (0.66) TTRMAPTHPGDNR1I2LMNA
Soneclosan SCHEMBL465591 0.86 TTR (0.66) TTRMAPTHPGDNR1I2LMNA
SCHEMBL10540653 0.85 TTR (0.83) TTRMAPTHPGDNR1I2LMNA
SCHEMBL14861327 0.84 TTR (0.50) TTRMAPTHPGDNR1I2LMNA
SCHEMBL10940178 0.82 CYP1A2 (0.62) TTRMAPTHPGDNR1I2LMNA
SCHEMBL29352050 0.82 CYP1A2 (0.62) TTRMAPTHPGDNR1I2LMNA
SCHEMBL11663615 0.80 CA1 (0.43) TTRMAPTHPGDNR1I2LMNA
SCHEMBL13778174 0.79 TTR (0.58) TTRMAPTHPGDNR1I2LMNA
SCHEMBL7182380 0.79 TTR (0.58) TTRMAPTHPGDNR1I2LMNA
SCHEMBL7176805 0.79 TTR (0.58) TTRMAPTHPGDNR1I2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 26 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1585751-A4 PEPTIDE DEFORMYLASE ACTIVATED PRODRUGS CELMED ONCOLOGY USA INC (CA) 2008-08-13 EP claimed
JP-2006514009-A 2006-04-27 JP claimed
US-20060063743-A1 Peptide deformylase activated prodrugs BALLATORE CARLO 2006-03-23 US claimed
EP-1585751-A2 PEPTIDE DEFORMYLASE ACTIVATED PRODRUGS Celmed Oncology (USA), Inc. (CA) 2005-10-19 EP claimed
US-20040236096-A1 Peptide deformylase activated prodrugs NEWBIOTICS, INC. 2004-11-25 US claimed
WO-2004043400-A2 PEPTIDE DEFORMYLASE ACTIVATED PRODRUGS CELMED ONCOLOGY (USA), INC. (CA) 2004-05-27 WO claimed
EP-1263762-A4 ANTI-INFECTIVE ECTATM NEWBIOTICS INC (US) 2003-04-02 EP claimed
EP-1263762-A1 ANTI-INFECTIVE ECTATM Newbiotics Inc. (US) 2002-12-11 EP claimed
WO-2001064687-A1 ANTI-INFECTIVE ECTA?TM¿ NEWBIOTICS, INC. (US) 2001-09-07 WO claimed
EP-1585751-A4 PEPTIDE DEFORMYLASE ACTIVATED PRODRUGS CELMED ONCOLOGY USA INC (CA) 2008-08-13 EP disclosed
US-7163923-B2 Bactericides, fungicides, viricides CELMED ONCOLOGY (USA), INC. (CA) 2007-01-16 US disclosed
EP-1499318-A4 PEPTIDE DEFORMYLASE ACTIVATED PRODRUGS CELMED ONCOLOGY USA INC (CA) 2006-07-19 EP disclosed
US-20060063743-A1 Peptide deformylase activated prodrugs BALLATORE CARLO 2006-03-23 US disclosed
US-7001922-B2 Peptide deformylase activated prodrugs CELMED ONCOLOGY (USA), INC. (CA) 2006-02-21 US disclosed
US-20030130179-A1 Methods for identifying therapeutic targets for treating infectious disease NEWBIOTICS, INC. 2003-07-10 US disclosed
US-20030091587-A1 Peptide deformylase activated prodrugs CELMED ONCOLOGY (USA), INC. (CA) 2003-05-15 US disclosed
EP-1263762-A4 ANTI-INFECTIVE ECTATM NEWBIOTICS INC (US) 2003-04-02 EP disclosed
EP-1263762-A1 ANTI-INFECTIVE ECTATM Newbiotics Inc. (US) 2002-12-11 EP disclosed
WO-2002007780-A2 METHODS FOR IDENTIFYING THERAPEUTIC TARGETS NEWBIOTICS, INC. (US) 2002-01-31 WO disclosed
WO-2001064687-A1 ANTI-INFECTIVE ECTA?TM¿ NEWBIOTICS, INC. (US) 2001-09-07 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060063743-A1 Peptide deformylase activated prodrugs DNPEP, DPEP1, PEPD TTR 3927/4885MAPT 4149/4885HPGD 732/4885
US-20040236096-A1 Peptide deformylase activated prodrugs DNPEP, DPEP1, PEPD TTR 4046/4885MAPT 4273/4885HPGD 850/4885
US-20030130179-A1 Methods for identifying therapeutic targets for treating infectious disease GAA, GBA3, RNASE1 TTR 3471/4885MAPT 3214/4885HPGD 851/4885
US-20030091587-A1 Peptide deformylase activated prodrugs DNPEP, PREP, DPEP1 TTR 3918/4885MAPT 4740/4885HPGD 360/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.