SCHEMBL4587399

SCHEMBL4587399

CCOC(=O)c1cnc2ccc(/C=C3\SC(Nc4cc(NC(=O)C(C)C)ccc4Cl)=NC3=O)cc2c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.38
SMN1; SMN2 Q16637 3/20 0.38
NPC1 O15118 2/20 0.38
RAB9A P51151 2/20 0.38
KMT2A Q03164 4/20 0.36
MEN1 O00255 3/20 0.36
CISD1 Q9NZ45 1/20 0.36
P2RY12 Q9H244 6/20 0.36
LMNA P02545 2/20 0.35
HPGD P15428 2/20 0.35
MITF O75030 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
IGF1R P08069 1/20 0.35
HDAC4 P56524 2/20 0.34
MAPT P10636 4/20 0.34
ABCB1 P08183 1/20 0.34
HTT P42858 1/20 0.34
ABCG2 Q9UNQ0 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL2995753 0.95 CISD1 (0.35) ALDH1A1SMN1; SMN2NPC1RAB9AKMT2A
Trifluoroacetic Acid SCHEMBL5050802 0.95 CISD1 (0.35) ALDH1A1SMN1; SMN2NPC1RAB9AKMT2A
SCHEMBL4586480 0.90 IGF1R (0.37) ALDH1A1SMN1; SMN2NPC1RAB9AKMT2A
SCHEMBL4586165 0.88 RAB9A (0.37) SMN1; SMN2NPC1RAB9AKMT2AMEN1
Trifluoroacetic Acid SCHEMBL2991044 0.84 DHODH (0.38) NPC1RAB9AKMT2AMEN1CISD1
Trifluoroacetic Acid SCHEMBL5049812 0.84 DHODH (0.38) NPC1RAB9AKMT2AMEN1CISD1
SCHEMBL2988361 0.83 SRC (0.39) ALDH1A1SMN1; SMN2KMT2AMEN1CISD1
SCHEMBL5049962 0.83 SRC (0.39) ALDH1A1SMN1; SMN2KMT2AMEN1CISD1
SCHEMBL2996481 0.83 DYRK3 (0.42) ALDH1A1NPC1RAB9AKMT2AMEN1
SCHEMBL2996479 0.83 DYRK3 (0.42) ALDH1A1NPC1RAB9AKMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1879563-A4 NOVEL CHEMICAL COMPOUNDS SMITHKLINE BEECHAM CORP (US) 2008-07-16 EP claimed
EP-1879563-A2 NOVEL CHEMICAL COMPOUNDS Smithkline Beecham Corporation (US) 2008-01-23 EP claimed
WO-2006132739-A2 NOVEL CHEMICAL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2006-12-14 WO claimed