SCHEMBL4587723

SCHEMBL4587723

FC(F)(F)c1cccc(C2CCN(CCc3ccc4ccoc4c3)CC2)c1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 3/20 0.57
DRD4 P21917 2/20 0.47
GRM2 Q14416 1/20 0.47
KDM4A O75164 1/20 0.46
KDM4B O94953 1/20 0.46
KDM5C P41229 1/20 0.46
KDM5B Q9UGL1 1/20 0.46
CHRM4 P08173 2/20 0.43
HTR2C P28335 2/20 0.42
HTR1A P08908 2/20 0.41
ALDH1A1 P00352 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
MAPT P10636 1/20 0.41
TSHR P16473 1/20 0.41
NFKB1 P19838 1/20 0.41
MAPK1 P28482 1/20 0.41
CYP2C19 P33261 1/20 0.41
THPO P40225 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9422688 0.84 DRD2 (0.63) DRD2DRD4GRM2KDM4AKDM4B
Hydrochloric Acid SCHEMBL9305904 0.83 DRD2 (0.62) DRD2DRD4GRM2KDM4AKDM4B
SCHEMBL4589239 0.80 DRD2 (0.57) DRD2DRD4GRM2KDM4AKDM4B
SCHEMBL9311321 0.79 DRD2 (0.66) DRD2DRD4GRM2KDM4AKDM4B
SCHEMBL1401478 0.79 DRD2 (0.56) DRD2DRD4GRM2KDM4AKDM4B
SCHEMBL1401365 0.79 DRD2 (0.56) DRD2DRD4GRM2KDM4AKDM4B
Hydrochloric Acid SCHEMBL4589565 0.78 DRD2 (0.55) DRD2DRD4GRM2KDM4AKDM4B
SCHEMBL1401419 0.77 DRD2 (0.60) DRD2DRD4GRM2KDM4AKDM4B
SCHEMBL4587366 0.77 DRD2 (0.56) DRD2DRD4GRM2KDM4AKDM4B
Hydrochloric Acid SCHEMBL1401480 0.76 DRD2 (0.58) DRD2DRD4GRM2KDM4AKDM4B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7326720-B2 Phenyl- and pyridylpiperidines with TNF activity SANOFI-AVENTIS (FR) 2008-02-05 US claimed